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4

抑制剂 & 化合物

10

天然产物

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Cat. No. Product Name Target Signaling Pathways
T15687 Thioflosulide

L-745337

COX Immunology/Inflammation; Neuroscience
Thioflosulide (L-745337) 是一种具有选择性和高效性的 COX2 抑制剂(IC50:2.3 nM),具有抗炎活性,可用于研究胃溃疡。
T68073 Flosatidil

Calcium Channel Membrane transporter/Ion channel; Metabolism
Flosatidil是一种小分子电压门控性钙通道复合体(VDCCs)阻滞剂,可用于治疗神经系统疾病和心血管疾病,可用于研究心绞痛。
T31805 Flosequinan

Others Others
Flosequinan 是一种动静脉血管扩张剂,已被证明可有效治疗急性心力衰竭。
T11296 Flosulide

ZK 38997,CGP 28238

COX Immunology/Inflammation; Neuroscience
Flosulide is an effective selective COX-2 inhibitor for the treatment of inflammatory diseases.

化合物

Thioflosulide
Cat.No: T15687
Synonym: L-745337
Target: COX
Flosatidil
Cat.No: T68073
Synonym:
Target: Calcium Channel
Flosequinan
Cat.No: T31805
Synonym:
Target: Others
Flosulide
Cat.No: T11296
Synonym: ZK 38997,CGP 28238
Target: COX
Cat. No. Product Name Target Signaling Pathways
T3858 macranthoidin A

灰毡毛忍冬皂苷甲,金银花

Others Others
Macranthoidin A 是一种具有口服活性的、提取于金银花中的皂苷。它对四氯化碳,对乙酰氨基酚和镉所致的肝损伤具有保护作用,对耳巴豆油的溶胀具有明显的抑制作用。
TN6556 Safflospermidine B

Safflospermidine B is a potential natural tyrosinase inhibitor, it shows high antityrosinase activity (IC50 of 31.8μM).
TN6555 Safflospermidine A

Safflospermidine A is a potential natural tyrosinase inhibitor,it shows high antityrosinase activity (IC50 of 13.8 μM).
TN4676 Nudifloside B

Others Others
Nudifloside B is a natural product from Jasminum nudiflorum.
TN4677 Nudifloside C

Others Others
Nudifloside C is a natural product from Jasminum nudiflorum.
TN4678 Nudifloside D

Others Others
Nudifloside D is a natural product from Jasminum nudiflorum.
T3367 Macranthoidin B

灰毡毛忍冬皂苷乙,金银花,Macranthoiside I

Others Others
Macranthoidin B (Macranthoiside I) 是一种活性天然皂苷。
T5787 Macranthoside B

金银花,灰毡毛忍冬次皂苷乙

Antibacterial Microbiology/Virology
Macranthoside B 是一种从金银花中分离出来的天然产物,具有抗菌活性。
TL0005 3,5-O-Dicaffeoylquinic acid

Isochlorogenic Acid A,(-)-3,5-二咖啡酰奎宁酸,(-)-3,5-Dicaffeoyl quinic acid,3,5-Dicaffeoylquinic Acid

Others Others
3,5-O-Dicaffeoylquinic acid (Isochlorogenic Acid A) 能够改善由三甲基锡诱导的学习和记忆缺陷。
T6S1294 Nicotiflorin

Nictoflorin,Kaempferol-3-O-Rutinoside,山奈酚-3-O-芸香糖苷,Nicotifloroside

Others Others
Nicotiflorin (Kaempferol-3-O-Rutinoside) 是一种黄酮苷,从传统中药Flos Carthami 中提取得到。它有抗糖化活性和神经保护作用。

天然产物

macranthoidin A
Cat.No: T3858
Synonym: 灰毡毛忍冬皂苷甲,金银花
Target: Others
Safflospermidine B
Cat.No: TN6556
Synonym:
Target:
Safflospermidine A
Cat.No: TN6555
Synonym:
Target:
Nudifloside B
Cat.No: TN4676
Synonym:
Target: Others
Nudifloside C
Cat.No: TN4677
Synonym:
Target: Others
Nudifloside D
Cat.No: TN4678
Synonym:
Target: Others
Macranthoidin B
Cat.No: T3367
Synonym: 灰毡毛忍冬皂苷乙,金银花,Macranthoiside I
Target: Others
Macranthoside B
Cat.No: T5787
Synonym: 金银花,灰毡毛忍冬次皂苷乙
Target: Antibacterial
3,5-O-Dicaffeoylquinic acid
Cat.No: TL0005
Synonym: Isochlorogenic Acid A,(-)-3,5-二咖啡酰奎宁酸,(-)-3,5-Dicaffeoyl quinic acid,3,5-Dicaffeoylquinic Acid
Target: Others
Nicotiflorin
Cat.No: T6S1294
Synonym: Nictoflorin,Kaempferol-3-O-Rutinoside,山奈酚-3-O-芸香糖苷,Nicotifloroside
Target: Others
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