Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2196 |
Fipronil
氟虫腈,Fluocyanobenpyrazole,Termidor |
P450; GluCls; GABA Receptor | Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience |
Fipronil (Fluocyanobenpyrazole) 是昆虫GABA 受体的选择性拮抗剂,可抑制蟑螂神经元中谷氨酸盐引起的脱敏和非脱敏。在分离的大鼠肝微粒体中,它诱导细胞色素 P450 (CYP) 亚型CYP1A1/2、CYP2B1/2和CYP3A1/2的活性。 | |||
T21071 |
Fipronil sulfone
|
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Fipronil sulfone is an insecticide fipronil. Its metabolite fipronil sulphone is an inhibitor of rat ɑ1β2γ2L GABA(A) receptor. | |||
T25428 |
Flufiprole
Rizazole,Butene-fipronil |
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Flufiprole is used as a phenylpyrazole pesticide. It has enantioselective metabolism in human and rat liver microsomes. |