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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T9926 | Omalizumab | Others | Others |
Omalizumab 是针对人免疫球蛋白 E 的重组人源化单克隆抗体(KD:0.393 nM)。它能够结合人 FcγRIIb 受体(KD:6.37 uM)。它对持续性过敏性哮喘具有潜在的研究价值。 | |||
T68689 | 2',3'-Dihydroxypuberulin | ||
2',3'-Dihydroxypuberulin is a natural inhibitor for FcεRI expression on mast cell from Verbasucum thapsus L. 2',3'-Dihydroxypuberulin was isolated from Pterocaulon balansae and P. lanatum. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN1154 |
Nepetin
6-Methoxyluteolin,泽兰黄酮,6-甲氧基藤黄菌素 |
Calcium Channel; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience |
Nepetin (6-Methoxyluteolin) 是一种分离自Eupatorium ballotaefoliumHBK 中的天然类黄酮,具有有效的抗炎作用。它在 ARPE-19 细胞中能够抑制IL-6(IC50:4.43 μM) 、IL-8 (IC50:43.42 μM) 、MCP-1 (IC50:4.17 μM) 的分泌。 |