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Cat. No. Product Name Target Signaling Pathways
T21653 1,4-DPCA

HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; Metabolism
1,4-DPCA 是一种脯氨酰羟化酶抑制剂,对人源包皮成纤维细胞中胶原羟基化的 IC50 为 2.4 μM,对因子抑制 HIF (FIH) 的 IC50 为 60 μM。
T1823 IOX2

IOX 2,JICL38

HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; Metabolism
IOX2 (IOX 2) 是特异性的脯氨酰羟化酶-2 抑制剂,IC50=22 nM。
T36796 1,4-DPCA ethyl ester

1,4-DPCA ethyl ester, the ethyl ester derivative of 1,4-DPCA, acts as an inhibitor of the enzyme factor inhibiting HIF (FIH)[1].
T68507 DM-NOFD

DM-NOFD is a cell penetrant prodrug of NOFD, which is a potent and selective inhibitor of an asparaginyl hydroxylase FIH (factor-inhibiting HIF).
T4651 Vadadustat

N-(5-(3-氯苯基)-3-羟基吡啶-2-羰基)甘氨酸,PG-1016548,AKB-6548

HIF/HIF Prolyl-Hydroxylase; HIF Angiogenesis; Chromatin/Epigenetic; Metabolism
Vadadustat 是一种可滴定口服的缺氧诱导因子脯氨酰羟化酶 (HIF-PH) 抑制剂,是一种促红细胞生成剂,在动物慢性肾脏疾病模型中,有用于贫血的研究潜力。

化合物

1,4-DPCA
Cat.No: T21653
Synonym:
Target: HIF/HIF Prolyl-Hydroxylase
IOX2
Cat.No: T1823
Synonym: IOX 2,JICL38
Target: HIF/HIF Prolyl-Hydroxylase
1,4-DPCA ethyl ester
Cat.No: T36796
Synonym:
Target:
DM-NOFD
Cat.No: T68507
Synonym:
Target:
Vadadustat
Cat.No: T4651
Synonym: N-(5-(3-氯苯基)-3-羟基吡啶-2-羰基)甘氨酸,PG-1016548,AKB-6548
Target: HIF/HIF Prolyl-Hydroxylase, HIF
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