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Cat. No. Product Name Target Signaling Pathways
T11282 FGTI-2734

Transferase Metabolism
FGTI-2734 是 有效的RAS C-末端法尼基转移酶 (FT) 和香叶烯基转移酶-1 (GGT-1) 抑制剂,IC50s 分别为 250 nM 和 520 nM。 它可以阻断 KRAS 的膜定位,从而解决 KRAS 耐药性问题,并抑制突变的 KRAS 胰腺肿瘤。
T11282L FGTI-2734 mesylate (1247018-19-4 free base)

FGTI-2734 mesylate

Others Others
FGTI-2734 mesylate, a RAS C-terminal mimetic compound with dual farnesyl transferase (FT) and geranylgeranyl transferase-1 (GGT) inhibitory activities (IC50s of 250 nM and 520 nM for FT and GGT, respectively), mitigates KRAS resistance by preventing its membrane localization, effectively impeding mutant KRAS patient-derived pancreatic tumors.

化合物

FGTI-2734
Cat.No: T11282
Synonym:
Target: Transferase
FGTI-2734 mesylate (1247018-19-4 free base)
Cat.No: T11282L
Synonym: FGTI-2734 mesylate
Target: Others
TargetMol Loading
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