Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T78832 |
FGFR1 inhibitor-9
|
FGFR | Angiogenesis; Tyrosine Kinase/Adaptors |
FGFR1inhibitor-9(Compound 9),一种FGFR1抑制剂(IC50为0.85 nM),可与FGFR1的ATP结合袋发生结合,并展现出抗癌活性。 | |||
T78831 |
FGFR1 inhibitor-8
|
FGFR | Angiogenesis; Tyrosine Kinase/Adaptors |
FGFR1inhibitor-8(化合物9)是一种高效的FGFR1抑制剂,其IC50s为0.5 nM,能够与FGFR1的ATP结合口袋发生相互作用,并显示出抗癌活性。 | |||
T39896 |
ALK-IN-9
|
||
ALK-IN-9 (compound 40) is a highly effective ALK inhibitor. It demonstrates remarkable inhibitory activity against cell proliferation, with IC50 values of <0.2 nM for Ba/F3-EML4-ALK, KM 12 (TPM3-TRKA), and KG-l cell (OP2-FGFR1). | |||
T73316 |
FGFR-IN-9
|
||
FGFR-IN-9 是一种有效的、可逆的、具有口服活性的FGFR 抑制剂,对FGFR4WT、FGFR3、FGFR4V550L、FGFR2 和FGFR1的IC50分别为 17.1、29.6、30.7、46.7 和 64.3 nM。 |