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Cat. No.	Product Name	Target	Signaling Pathways
T9855	BR102910 4-Thiazolecarboxamide, N-[2-[(2S)-2-cyano-4,4-difluoro-1-pyrrolidinyl]-2-oxoethyl]-2-[(3,4-dichlorophenyl)methyl]-	Others	Others
	BR102910 (4-Thiazolecarboxamide, N-[2-[(2S)-2-cyano-4,4-difluoro-1-pyrrolidinyl]-2-oxoethyl]-2-[(3,4-dichlorophenyl)methyl]-) 是一种选择性的成纤维细胞活化蛋白（FAP）的抑制剂。
T7890	SP-13786 UAMC-1110,(S)-N-[2-(2-氰基-4,4-二氟-1-吡咯烷基)-2-氧代乙基]喹啉-4-甲酰胺	Others	Others
	SP-13786 (UAMC-1110) 是成纤维细胞活化蛋白 (FAP) 的抑制剂 (IC50 : 3.2 nM)；还抑制脯氨酰寡肽酶 (PREP) ( IC50 : 1.8 μM)。
T78214	FAP-IN-2 TFA
	FAP-IN-2 TFA为99mTc标记的异腈类FAP抑制剂衍生物，适用于肿瘤显像。
T11263	FAPI-2	Others	Others
	Fapi-2 is a fibroblast activated protein (FAP) inhibitor used in cancer research.
T35852	FAPI-34
	FAPI-34, a fibroblast-activating protein (FAP) inhibitor, boasts advantageous pharmacokinetic and biochemical attributes.
T10227	Ac-Gly-BoroPro	Others	Others
	Ac-Gly-BoroPro is a selective FAP inhibitor (Ki: 23 nM).
T69603	BR103354
	BR103354 is a novel fibroblast activation protein (FAP) inhibitor with anti-diabetic and anti-steatotic effects. BR103354 inhibited FAP with an IC50 value of 14 nM, showing high selectivity against dipeptidyl peptidase (DPP)-related enzymes and prolyl oligopeptidase (PREP). BR103354 exhibited good pharmacokinetic properties as evidenced by oral bioavailability of 48.4% and minimal hERG inhibition. Single co-administration of BR103354 with hFGF21 reduced nonfasting blood glucose concentrations, i...
T11264	FAPI-4	Others	Others
	Api-4 is a fibroblast activated protein (FAP) inhibitor used in cancer research.
T78921	FAP-IN-1
	FAP-IN-1，一种FAP (成纤维细胞激活蛋白)抑制剂，具有3.3 nM的IC50值，适用于癌症研究。
T74402	FAP-PI3KI1
	FAP-PI3KI1 是一种成纤维细胞活化蛋白 (FAP) 靶向 PI3K 抑制剂，可选择性靶向表达 FAP 的人特发性肺纤维化 (IPF)细胞并有效抑制胶原蛋白合成，减少胶原蛋白沉积。
T82416	FAPI-2 TFA
	FAPI-2 TFA为一种针对成纤维细胞活化蛋白（FAP）的抑制剂，适用于癌症研究领域。
T69660	NOTA-FAPI-4
	NOTA-FAPI-4 is an analogue of FAPI-4 and a fibroblast activation protein (FAP) inhibitor. NOTA-FAPI-4 is useful in the diagnosis or treatment of a disease characterized by overexpression of fibroblast activation protein (FAP). NOTA-FAPI-4 can be used as a PET tracer for detection of diseases or disorders related to fibroblast activation protein.
T79917	FAP-IN-2
	FAP-IN-2，一种标记有99mTc的含异腈FAPI（成纤维细胞活化蛋白）抑制剂衍生物，适用于肿瘤显像。
T78179	NH2-UAMC1110 TFA
	NH2-UAMC1110 TFA 是 UAMC1110 的一个衍生物，用于合成 FAPI-QS。UAMC1110 是成纤维细胞激活蛋白（FAP）的抑制剂，而 FAPI-QS 作为螯合剂，用于制备特异性高、剂量大的放射性示踪剂，适用于肿瘤的诊断与治疗。
T37861	Talabostat
	Talabostat (PT100, Val-boroPro) is a potent, nonselective and orally available dipeptidyl peptidase IV (DPP-IV) inhibitor with a Ki of 0.18 nM. Talabostat is a nonselective DPP-IV inhibitor, inhibiting DPP8/9, FAP, DPP2 and some other DASH family enzymes essentially as potently as it inhibits DPP-IV[1]. Talabostat stimulates the immune system by triggering a proinflammatory form of cell death in monocytes and macrophages known as pyroptosis. The inhibition of two serine proteases, DPP8 and DPP9,...

化合物

Cat.No: T9855

Synonym: 4-Thiazolecarboxamide, N-[2-[(2S)-2-cyano-4,4-difluoro-1-pyrrolidinyl]-2-oxoethyl]-2-[(3,4-dichlorophenyl)methyl]-

Target: Others

Cat.No: T7890

Synonym: UAMC-1110,(S)-N-[2-(2-氰基-4,4-二氟-1-吡咯烷基)-2-氧代乙基]喹啉-4-甲酰胺

Target: Others

Cat.No: T78214

Cat.No: T11263

Target: Others

Cat.No: T35852

Cat.No: T10227

Target: Others

Cat.No: T69603

Cat.No: T11264

Target: Others

Cat.No: T78921

Cat.No: T74402

Cat.No: T82416

Cat.No: T69660

Cat.No: T79917

NH2-UAMC1110 TFA

Cat.No: T78179

Cat.No: T37861

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