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Cat. No. Product Name Target Signaling Pathways
T0373L Erlotinib hydrochloride

盐酸埃罗替尼,OSI-744,NSC 718781,Erlotinib HCl,CP-358774

EGFR; Autophagy Angiogenesis; Autophagy; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Erlotinib hydrochloride (NSC 718781) 抑制EGFR 激酶的IC50为 2 nM,用于治疗非小细胞肺癌。
T6619 Desmethyl Erlotinib hydrochloride

OSI420,OSI-420,DesMethyl Erlotinib (CP-473420) HCl,去甲厄洛替尼,CP-473420,Desmethyl Erlotinib,OSI 420

EGFR; Drug Metabolite Angiogenesis; JAK/STAT signaling; Metabolism; Tyrosine Kinase/Adaptors
Desmethyl Erlotinib hydrochloride (OSI 420) 是 Erlotinib 的活性代谢物。Erlotinib 是 EGFR 酪氨酸激酶抑制剂。
T19312 Erlotinib-d6 hydrochloride

CP-358774 D6 hydrochloride,NSC 718781 D6 hydrochloride,Erlotinib D6 hydrochloride,OSI-774 D6 hydrochloride

Others Others
Erlotinib Hydrochloride inhibits purified EGFR kinase with an IC50 of 2 nM. Erlotinib D6 hydrochloride a deuterium labeled Erlotinib Hydrochloride.

化合物

Erlotinib hydrochloride
Cat.No: T0373L
Synonym: 盐酸埃罗替尼,OSI-744,NSC 718781,Erlotinib HCl,CP-358774
Target: EGFR, Autophagy
Desmethyl Erlotinib hydrochloride
Cat.No: T6619
Synonym: OSI420,OSI-420,DesMethyl Erlotinib (CP-473420) HCl,去甲厄洛替尼,CP-473420,Desmethyl Erlotinib,OSI 420
Target: EGFR, Drug Metabolite
Erlotinib-d6 hydrochloride
Cat.No: T19312
Synonym: CP-358774 D6 hydrochloride,NSC 718781 D6 hydrochloride,Erlotinib D6 hydrochloride,OSI-774 D6 hydrochloride
Target: Others
TargetMol Loading
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