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Cat. No. Product Name Target Signaling Pathways
T6075 Epothilone B

帕妥匹隆,Patupilone,EPO 906

Apoptosis; Microtubule Associated; Antibiotic; Antifungal Apoptosis; Cytoskeletal Signaling; Microbiology/Virology
Epothilone B (EPO 906) 是微管稳定剂,Ki 为0.71 μM。 它与αβ-微管蛋白异二聚体亚基结合,使αβ-微管蛋白解离减少。
T6864 Ixabepilone

BMS 247550,Ixempra,Azaepothilone B,伊沙匹隆,BMS 247550-1

Apoptosis; Microtubule Associated Apoptosis; Cytoskeletal Signaling
Ixabepilone (Azaepothilone B) 是一种可口服的微管抑制剂,能够与微管蛋白结合,促进微管蛋白的聚合和微管的稳定,使细胞停滞在 G2-M 期,诱导细胞凋亡。
T73084 BMS 310705

21-Aminoepothilone B

BMS 310705 (21-Aminoepothilone B) 是 Epothilone B 的类似物,靶向卵巢癌、肾癌、膀胱癌和肺癌等恶性肿瘤。BMS 310705 通过线粒体介导的途径诱导显着的细胞凋亡 (apoptosis)。
T68860 Iso-Fludelone

Iso-Fludelone is the third-generation epothilone B analogue with potential anti-mitotic and antineoplastic activites. Iso-fludelone binds to tubulin and induces microtubule polymerization and stabilizes microtubules against depolymerization, which may result in the inhibition of cell division, the induction of G2/M arrest, and apoptosis. Compared to other generations of epothilones, iso-fludelone exhibits increased stability, water solubility, potency, duration of action, tumor penetration as we...

化合物

Epothilone B
Cat.No: T6075
Synonym: 帕妥匹隆,Patupilone,EPO 906
Target: Apoptosis, Microtubule Associated, Antibiotic, Antifungal
Ixabepilone
Cat.No: T6864
Synonym: BMS 247550,Ixempra,Azaepothilone B,伊沙匹隆,BMS 247550-1
Target: Apoptosis, Microtubule Associated
BMS 310705
Cat.No: T73084
Synonym: 21-Aminoepothilone B
Target:
Iso-Fludelone
Cat.No: T68860
Synonym:
Target:
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