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10

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T69109 Ellipticine tartrate

Ellipticine tartrate is a DNA intercalating agent and a DNA topoisomerase II inhibitor.
T68788 Ellipticine quinone

Ellipticine quinone, also known as NSC-383230, is a Drp1 inhibitor. rpitor1 and Drpitor1a inhibited the GTPase activity of Drp1 without inhibiting the GTPase of dynamin 1. Ellipticine quinone showed greater potency than the current std. Drp1 GTPase inhibitor, mdivi-​1, (IC50 for mitochondrial fragmentation are (0.06, and 10 μM, resp.)​. Ellipticine quinone suppressed lung cancer tumor growth in a mouse xenograft model. Ellipticine quinone also inhibited mitochondrial ROS prodn., prevented mi...
T82560 di-Ellipticine-RIBOTAC

PROTACs PROTAC
Di-Ellipticine-RIBOTAC是一款双功能小分子,在体外和体内肌萎缩侧索硬化(ALS)模型中能够减少c9ALS/FTD r(G4C2)的重复扩增。
T7747 Datelliptium chloride hydrochloride

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Datelliptium chloride hydrochloride 是一种衍生自玫瑰树碱的 DNA 嵌入剂,具有抗肿瘤活性。
T36699 9-Methoxyellipticine

9-Methoxyellipticine is an alkaloid and a derivative of the DNA intercalating agent ellipticine that has been found in O. maculataand has anticancer activity.It intercalates into DNA and is an inhibitor of wild-type c-Kit and c-Kit containing the D816V activating mutation (c-KitD816V; IC50s = 0.8 and 0.6 μM, respectively).
T27562 Hydroxyellipticine-1a

Hydroxyellipticine-1a, a selective r(CGG)exp probe, improves pre-mRNA splicing defects, inhibits formation of nuclear inclusions and RANT in a FXTAS cellular mode.l
T10200 9-Hydroxyellipticine hydrochloride

Others Others
9-Hydroxyellipticine hydrochloride is a inhibitor of Topo II and RyR. It exhibits antitumor, antioxidant and catecholamine-releasing activities. 9-Hydroxyellipticine hydrochloride inihibits Hela S-3 and 293T cells (IC50s: 1.6 μM and 1.2μM).
T26401 9-Hydroxyellipticin free base

IGIG929,NSC 210717,9-hydroxyellipticine,IGIG 929,9-Hydroxyellipticin,Hydroxyellipticine

9-hydroxyellipticine is a potent cytotoxic and antitumor agent. 9-hydroxyellipticine is a 9-hydroxy derivative of ellipticine.
T7429 Datelliptium chloride

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Datelliptium chloride 是一种源自玫瑰树碱的 DNA 嵌入剂,具有抗肿瘤活性。
T41151 K34c

K34c is a potent and selective α5β1 integrin inhibitor (IC50 = 3.1 nM). K34c inhibits cell survival and migration, inhibits p53-dependent senescence induced by Temozolomide or Ellipticine and promotes apoptosis in U87MG cells. K34c also prevents TGFβ-induced infiltrationin vivoand reduces cell adhesion on fibronectin.

化合物

Ellipticine tartrate
Cat.No: T69109
Synonym:
Target:
Ellipticine quinone
Cat.No: T68788
Synonym:
Target:
di-Ellipticine-RIBOTAC
Cat.No: T82560
Synonym:
Target: PROTACs
Datelliptium chloride hydrochloride
Cat.No: T7747
Synonym:
Target: DNA/RNA Synthesis
9-Methoxyellipticine
Cat.No: T36699
Synonym:
Target:
Hydroxyellipticine-1a
Cat.No: T27562
Synonym:
Target:
9-Hydroxyellipticine hydrochloride
Cat.No: T10200
Synonym:
Target: Others
9-Hydroxyellipticin free base
Cat.No: T26401
Synonym: IGIG929,NSC 210717,9-hydroxyellipticine,IGIG 929,9-Hydroxyellipticin,Hydroxyellipticine
Target:
Datelliptium chloride
Cat.No: T7429
Synonym:
Target: DNA/RNA Synthesis
K34c
Cat.No: T41151
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1166 Ellipticine

玫瑰树碱,NSC 71795,Elliptisine

Topoisomerase DNA Damage/DNA Repair
Ellipticine (Elliptisine) 是一种有效的抗肿瘤剂,抑制 DNA 拓扑异构酶 II 活性,对白血病、神经母细胞瘤和胶质母细胞瘤有部分活性。
T4614 Ellipticine hydrochloride

Ellipticine HCl,NSC 71795 (hydrochloride),玫瑰树碱盐酸盐

Topoisomerase DNA Damage/DNA Repair
Ellipticine hydrochloride (NSC-71795 (hydrochloride)) 是一种有效的抗肿瘤剂,抑制 DNA 拓扑异构酶 II 的活性。

天然产物

Ellipticine
Cat.No: T1166
Synonym: 玫瑰树碱,NSC 71795,Elliptisine
Target: Topoisomerase
Ellipticine hydrochloride
Cat.No: T4614
Synonym: Ellipticine HCl,NSC 71795 (hydrochloride),玫瑰树碱盐酸盐
Target: Topoisomerase
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