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Cat. No. Product Name Target Signaling Pathways
T1788 Tazemetostat

E-7438,EPZ6438

Histone Methyltransferase Chromatin/Epigenetic
Tazemetostat (EPZ6438) 是一种组蛋白甲基转移酶 EZH2 抑制剂 (IC50=11 nM),具有口服活性、选择性和 SAM 竞争性。Tazemetostat 具有抗肿瘤活性,可以用于治疗上皮样肉瘤/滤泡性淋巴瘤。
T17002 Tazemetostat hydrobromide

E-7438 hydrobromide,氢溴酸泰泽司他,EPZ-6438 hydrobromide

Histone Methyltransferase Chromatin/Epigenetic
Tazemetostat hydrobromide (E-7438 hydrobromide) 是口服的EZH2选择性抑制剂。它抑制含有 PRC2 复合体的野生型 EZH2 的活性,Ki 为 2.5 nM。它还抑制 EZH1,IC50为 392 nM。
T15240 Tazemetostat trihydrochloride

EPZ-6438 trihydrochloride,E-7438 trihydrochloride

Histone Methyltransferase Chromatin/Epigenetic
Tazemetostat trihydrochloride is a selective and orally available inhibitor of EZH2 (IC50: 4 nM for rat EZH2). It inhibits the activity of human PRC2-containing wild-type EZH2 (Ki: 2.5 nM). It inhibits EZH2 (IC50s: 11 and 16 nM in peptide assay and nucleo

化合物

Tazemetostat
Cat.No: T1788
Synonym: E-7438,EPZ6438
Target: Histone Methyltransferase
Tazemetostat hydrobromide
Cat.No: T17002
Synonym: E-7438 hydrobromide,氢溴酸泰泽司他,EPZ-6438 hydrobromide
Target: Histone Methyltransferase
Tazemetostat trihydrochloride
Cat.No: T15240
Synonym: EPZ-6438 trihydrochloride,E-7438 trihydrochloride
Target: Histone Methyltransferase
TargetMol Loading
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