Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6037 |
E-64
Proteinase inhibitor E 64,E 64,E64 |
Cysteine Protease; Antibacterial; Autophagy | Autophagy; Microbiology/Virology; Proteases/Proteasome |
E-64 (Proteinase inhibitor E 64)是一种不可逆的半胱氨酸蛋白酶抑制剂,抑制papain 的IC50为 9 nM。 | |||
T4068 |
E6446 dihydrochloride
|
TLR | Immunology/Inflammation |
E6446 dihydrochloride 是一种新型合成拮抗剂,用于核酸感应 TLR;有效抑制对 HEK:TLR9 细胞的 DNA 刺激,IC50 为 10 nM。 | |||
T4206 |
E6446
|
TLR | Immunology/Inflammation |
E6446 抑制 Toll 样受体 (TLR)7 和 9 信号传导。 E6446 在多种人和小鼠细胞类型中起作用,并在体外抑制 DNA-TLR9 相互作用。当给予小鼠时,该化合物抑制对刺激 TLR9 的含有胞苷-磷酸-胍 (CpG) 的 DNA 的挑战剂量的反应。 | |||
T11141 |
E64FC26
|
Others | Others |
E64FC26 是一种有效的蛋白质二硫键异构酶 (PDI) 家族泛抑制剂,具有抗肿瘤活性,抑制 PDIA1、PDIA3、PDIA4、TXNDC5 和 PDIA6,可用于研究多发性骨髓瘤和胰腺癌。 | |||
T39812 |
(E/Z)-E64FC26
(E/Z)-E64FC26 |
||
(E/Z)-E64FC26 is a mixture complex comprising E-E64FC26 and Z-E64FC26. E-E64FC26 is a highly potent pan-inhibitor of the protein disulfide isomerase (PDI) family, with IC50 values of 1.9, 20.9, 25.9, 16.3, and 25.4 μM against PDIA1, PDIA3, PDIA4, TXNDC5, and PDIA6, respectively. Furthermore, E64FC26 demonstrates anti-myeloma activity. | |||
T90016 |
Compound E643-0199
|
||
T90102 |
Compound E642-1065
|
||
T90201 |
Compound E641-1273
|
||
T90117 | Compound E642-1130 | ||
T90114 |
Compound E642-0521
|
||
T90202 |
Compound E641-1450
|
||
T90203 |
Compound E642-0876
|
||