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Cat. No. Product Name Target Signaling Pathways
T6037 E-64

Proteinase inhibitor E 64,E 64,E64

Cysteine Protease; Antibacterial; Autophagy Autophagy; Microbiology/Virology; Proteases/Proteasome
E-64 (Proteinase inhibitor E 64)是一种不可逆的半胱氨酸蛋白酶抑制剂,抑制papain 的IC50为 9 nM。
T4068 E6446 dihydrochloride

TLR Immunology/Inflammation
E6446 dihydrochloride 是一种新型合成拮抗剂,用于核酸感应 TLR;有效抑制对 HEK:TLR9 细胞的 DNA 刺激,IC50 为 10 nM。
T4206 E6446

TLR Immunology/Inflammation
E6446 抑制 Toll 样受体 (TLR)7 和 9 信号传导。 E6446 在多种人和小鼠细胞类型中起作用,并在体外抑制 DNA-TLR9 相互作用。当给予小鼠时,该化合物抑制对刺激 TLR9 的含有胞苷-磷酸-胍 (CpG) 的 DNA 的挑战剂量的反应。
T11141 E64FC26

Others Others
E64FC26 是一种有效的蛋白质二硫键异构酶 (PDI) 家族泛抑制剂,具有抗肿瘤活性,抑制 PDIA1、PDIA3、PDIA4、TXNDC5 和 PDIA6,可用于研究多发性骨髓瘤和胰腺癌。
T39812 (E/Z)-E64FC26

(E/Z)-E64FC26

(E/Z)-E64FC26 is a mixture complex comprising E-E64FC26 and Z-E64FC26. E-E64FC26 is a highly potent pan-inhibitor of the protein disulfide isomerase (PDI) family, with IC50 values of 1.9, 20.9, 25.9, 16.3, and 25.4 μM against PDIA1, PDIA3, PDIA4, TXNDC5, and PDIA6, respectively. Furthermore, E64FC26 demonstrates anti-myeloma activity.
T90016 Compound E643-0199

T90102 Compound E642-1065

T90201 Compound E641-1273

T90117 Compound E642-1130

T90114 Compound E642-0521

T90202 Compound E641-1450

T90203 Compound E642-0876

化合物

E-64
Cat.No: T6037
Synonym: Proteinase inhibitor E 64,E 64,E64
Target: Cysteine Protease, Antibacterial, Autophagy
E6446 dihydrochloride
Cat.No: T4068
Synonym:
Target: TLR
E6446
Cat.No: T4206
Synonym:
Target: TLR
E64FC26
Cat.No: T11141
Synonym:
Target: Others
(E/Z)-E64FC26
Cat.No: T39812
Synonym: (E/Z)-E64FC26
Target:
Compound E643-0199
Cat.No: T90016
Synonym:
Target:
Compound E642-1065
Cat.No: T90102
Synonym:
Target:
Compound E641-1273
Cat.No: T90201
Synonym:
Target:
Compound E642-1130
Cat.No: T90117
Synonym:
Target:
Compound E642-0521
Cat.No: T90114
Synonym:
Target:
Compound E641-1450
Cat.No: T90202
Synonym:
Target:
Compound E642-0876
Cat.No: T90203
Synonym:
Target:
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