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Cat. No. Product Name Target Signaling Pathways
T16078 Mirk-IN-1

Dyrk1B/A-IN-1

Others Others
Mirk-IN-1 is an effective inhibitor of Dyrk1B(Mirk kianse) and Dyrk1A (IC50: 68±48 nM and 22±8 nM respectively).
T11132 DYRKs-IN-1

DYRK Cell Cycle/Checkpoint; Tyrosine Kinase/Adaptors
DYRKs-IN-1 has antitumor activity. DYRKs-IN-1 is a potent DYRKs (Dual-specificity tyrosine-phosphorylation-regulated kinases) inhibitor with IC50s of 9 nM and 5 nM for DYRK1B and DYRK1A, respectively.
T62043 Dyrk1A/B-IN-1

Dyrk1A/B-IN-1 (compound 3n) 是有效的、选择性的和细胞渗透性的DYRK1ADYRK1B 抑制剂。Dyrk1A/B-IN-1抑制DYRK1ADYRK1B 的Ki 分别为 67.8 nM 和 237.9 nM,IC50分别为 1.1 μM 和 0.8 μM。
T72242 DYRKs-IN-1 hydrochloride

DYRKs-IN-1 hydrochloride是一种有效的DYRKs(双特异性酪氨酸磷酸化调节激酶)抑制剂,对DYRK1ADYRK1B的IC50分别为5 nM和8 nM,具有抗肿瘤活性。

化合物

Mirk-IN-1
Cat.No: T16078
Synonym: Dyrk1B/A-IN-1
Target: Others
DYRKs-IN-1
Cat.No: T11132
Synonym:
Target: DYRK
Dyrk1A/B-IN-1
Cat.No: T62043
Synonym:
Target:
DYRKs-IN-1 hydrochloride
Cat.No: T72242
Synonym:
Target:
TargetMol Loading
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