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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T36408 Rhein-13C4

Rhein-13C4

Rhein-13C4 is intended for use as an internal standard for the quantification of rhein by GC- or LC-MS. Rhein is an anti-inflammatory anthraquinone found in rhubarb and is the bioactive derivative of its prodrug diacerein . At 10 μM, rhein inhibits IL-1β signaling, suppressing signaling through NF-κB, and reduces the expression of the matrix metalloproteases MMP-1 and MMP-13.1 It inhibits IKKβ (IC50 = 11.8 μM), decreasing iNOS and IL-6 expression in LPS-stimulated macrophages but paradoxically i...

化合物

Rhein-13C4
Cat.No: T36408
Synonym: Rhein-13C4
Target:
Cat. No. Product Name Target Signaling Pathways
T1273 Diacerein

双醋瑞因,Diacerhein,Fisiodar,Diacetylrhein

IL Receptor; Interleukin Immunology/Inflammation
Diacerein (Fisiodar) 是一种慢效具有白介素-1β 抑制效果的蒽醌类化合物。
T2997 Rhein

Rheinic Acid,Monorhein,大黄酸,NSC 38629,Rheic Acid,Rhubarb yellow

Reactive Oxygen Species; Antibacterial; Autophagy Autophagy; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Rhein (NSC 38629) 从蓼科大黄中提取的一种蒽醌类化合物,有抗炎、抗氧化、抗癌等作用。

天然产物

Diacerein
Cat.No: T1273
Synonym: 双醋瑞因,Diacerhein,Fisiodar,Diacetylrhein
Target: IL Receptor, Interleukin
Rhein
Cat.No: T2997
Synonym: Rheinic Acid,Monorhein,大黄酸,NSC 38629,Rheic Acid,Rhubarb yellow
Target: Reactive Oxygen Species, Antibacterial, Autophagy
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