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1
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T79920 |
Debrisoquin
Debrisoquine,Ro 5-3307/1,Isocaramidine |
SARS-CoV | Microbiology/Virology |
Debrisoquin (Isocaramidine) 是一种抑制剂,针对TMPRSS2,能够在依赖TMPRSS2的机制中抑制SARS-CoV-2进入人肺细胞系,IC50 值为22 μM。该化合物适用于抗病毒研究领域。 | |||
T31272 |
Debrisoquin sulfate
Tendor,Isocaramidine,Debrisochinum,Debrisoquine,Debrisoquin,Debrisoquina |
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Debrisoquine is an antihypertensive drug similar to guanethidine. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TMA2106 | (-)-Sparteine | P450 | Metabolism |
Sparteine is a class 1a antiarrhythmic agent, a sodium channel blocker. The deficient debrisoquine hydroxylation of Sparteine is due to the absence of P-450IID1 protein in the livers of poor metabolizers. |