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Cat. No.	Product Name	Target	Signaling Pathways
T3337	Ddr1-In-1	Discoidin Domain Receptor (DDR)	Tyrosine Kinase/Adaptors
	DDR1-IN-1 是一种特异性的 DDR1 受体酪氨酸激酶抑制剂，选择性是 DDR2 的 3 倍左右。
T5402	DDR1-IN-2 DDR1 inhibitor 7rh	Discoidin Domain Receptor (DDR)	Tyrosine Kinase/Adaptors
	DDR1-IN-2 (DDR1 inhibitor 7rh) 是盘状结构域受体 1 抑制剂 (IC50:13.1 nM)，对 DDR2 的抑制作用相对较弱 (IC50:203 nM)。
T70202	DDR1-IN-1 dihydrochloride
	DDR1-IN-1 dihydrochloride 是 DDR1受体酪氨酸激酶抑制剂，IC50值为105 nM，而对 DDR2的 IC50为413 nM。
T70201	S 16020-2
	S 16020-2 is an olivacine derivative, and DNA topoisomerase II inhibitor endowed with a remarkable antitumor activity against various experimental tumors.
T39572	DDR1-IN-4 DDR1-IN-4
	DDR1-IN-4 (Compound 2.45) is a highly potent inhibitor that selectively targets Discoidin Domain Receptor 1 (DDR1) autophosphorylation. This compound demonstrates exceptional efficacy with IC50 values of 29 nM and 1.9 μM for DDR1 and DDR2, respectively.
T40062	DDR1-IN-5 DDR1-IN-5
	DDR1-IN-5 is a potent and selective inhibitor of the Discoidin Domain Receptor family, member 1 (DDR1). It effectively inhibits the phosphorylation of DDR1b (Y513) with an IC 50 value of 4.1 nM. Furthermore, DDR1-IN-5 demonstrates remarkable anti-cancer activity. Its inhibitory potency against DDR1 (IC 50 = 7.36 nM) makes it a promising compound for targeted therapy in cancer treatment.
T40061	DDR1-IN-6 DDR1-IN-6
	DDR1-IN-6 is a potent and selective inhibitor of Discoidin Domain Receptor family member 1 (DDR1), exhibiting remarkable inhibitory activity at an IC50 of 9.72 nM. It effectively suppresses the auto-phosphorylation of DDR1b (Y513) with an IC50 value of 9.7 nM. Furthermore, DDR1-IN-6 displays strong anti-cancer activity.
T79811	DDR1/2 inhibitor-2
	DDR1/2 inhibitor-2 (Example 31)，作为一种DDR1/DDR2抑制剂，其IC50值小于100 nM，适用于癌症和纤维化疾病的研究领域。

化合物

Cat.No: T3337

Target: Discoidin Domain Receptor (DDR)

Cat.No: T5402

Synonym: DDR1 inhibitor 7rh

Target: Discoidin Domain Receptor (DDR)

DDR1-IN-1 dihydrochloride

Cat.No: T70202

Cat.No: T70201

Cat.No: T39572

Synonym: DDR1-IN-4

Cat.No: T40062

Synonym: DDR1-IN-5

Cat.No: T40061

Synonym: DDR1-IN-6

DDR1/2 inhibitor-2

Cat.No: T79811

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