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3

抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T27116 D(-)-Octopamine CSA salt

D(-)-Octopamine CSA salt is an agonist of octopamine receptors.
T71508 TCSA

TCSA is an inhibitor of fungal morphogenesis, biofilm formation, and host cell invasion.
T34999 UNIL-088

UNIL 088

UNIL088 is a water-soluble prodrug of cyclosporine A (CsA) designed for topical ocular delivery. The pro-moiety is grafted via an ester function to CsA and the solubilizing group is a phosphate ion. UNIL-088 can be rapidly hydrolysed under physiological c

化合物

D(-)-Octopamine CSA salt
Cat.No: T27116
Synonym:
Target:
TCSA
Cat.No: T71508
Synonym:
Target:
UNIL-088
Cat.No: T34999
Synonym: UNIL 088
Target:
Cat. No. Product Name Target Signaling Pathways
T0945 Cyclosporin A

环孢素,Cyclosporine A,Ciclosporin,Cyclosporine,环孢菌素

Phosphatase; Antibiotic; Complement System Immunology/Inflammation; Metabolism; Microbiology/Virology
Cyclosporin A 属于天然产物,是一种真菌的活性代谢产物,一种环状多肽。Cyclosporin A 是一种能与亲环素结合的免疫抑制剂,可以抑制 calcineurin (IC50=7 nM)。

天然产物

Cyclosporin A
Cat.No: T0945
Synonym: 环孢素,Cyclosporine A,Ciclosporin,Cyclosporine,环孢菌素
Target: Phosphatase, Antibiotic, Complement System
TargetMol Loading
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