Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1247 |
Clonidine hydrochloride
Clonidine HCl,Catapres,盐酸可乐定 |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Clonidine hydrochloride (Catapres) 是一种α2-adrenoceptor 激动剂,是一种抗高血压药。 | |||
T40869 |
Moxonidine hydrochloride
BDF5895hydrochloride,盐酸莫索尼定 |
||
Moxonidine Hydrochloride is a selective agonist at the imidazoline receptor subtype 1, used as antihypertensive agent. Target: I1-R Moxonidine Hydrochloride is a centrally acting antihypertensive agent. Mixed Nischarin (I1 imidazoline receptor) and α2-AR (adrenergic) agonist; displays 40-fold higher affinity for I1 receptors versus α2-adrenoceptors. Moxonidine reduced stimulated NE overflow (log EC50: -6.15 +/- 0.14). AGN192403, a selective ligand at I1-R, had no influence on the dose-response... |