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Cat. No. Product Name Target Signaling Pathways
T5443 JQ-1 (carboxylic acid)

JQ-1 carboxylic acid

Epigenetic Reader Domain Chromatin/Epigenetic
JQ-1 (carboxylic acid) 是一种细胞渗透性 BRD4 抑制剂,对 BRD4(1) 和 BRD4(2) 的 IC50 分别为 77 和 33 nM。它是一种 (+)-JQ1 衍生物,可作为合成 PROTACs 的前体。
T15784 LP99

Epigenetic Reader Domain Chromatin/Epigenetic
LP99 是一种表观遗传探针,可破坏 BRD7 和 BRD9 与细胞中染色质的结合。它是一种选择性的 BRD7 和 BRD9 溴结构域抑制剂,对 BRD9 的 Kd 为 99 nM。
T39810 CEM114

CEM114 is a potent chemical compound known as a chemical epigenetic modifier (CEM). It functions by employing CRISPR-Cas9 systems to harness endogenous chromatin machinery, thereby exerting its epigenetic modifying effects.
T72013 Epigenetic Multiple Ligand

Epigenetic Multiple Ligand is a cell-permeable inhibitor of substrate processing by several chromatin-associated enzymes, including SIRT1/2, H3/SET7, H3/p300/CBP, H4/RmtA, PABP1/CARM1, and H4/PRMT1. It acts by inducing either apoptosis or granulocytic differentiation.

化合物

JQ-1 (carboxylic acid)
Cat.No: T5443
Synonym: JQ-1 carboxylic acid
Target: Epigenetic Reader Domain
LP99
Cat.No: T15784
Synonym:
Target: Epigenetic Reader Domain
CEM114
Cat.No: T39810
Synonym:
Target:
Epigenetic Multiple Ligand
Cat.No: T72013
Synonym:
Target:
TargetMol Loading
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