Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T14927 |
Centrinone
LCR-263 |
PLK; Aurora Kinase | Cell Cycle/Checkpoint; Chromatin/Epigenetic |
Centrinone (LCR-263) 是 polo 样激酶 4 的可逆抑制剂,对PLK4的Ki 值为0.16 nM。 | |||
T14926 |
Centrinone-B
LCR-323 |
Aurora Kinase | Cell Cycle/Checkpoint; Chromatin/Epigenetic |
Centrinone-B (LCR-323) is a potent and highly selective inhibitor of PLK4 (Ki: 0.59 nM). |