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Search Results for " carboxypeptidase inhibitor "

14

抑制剂 & 化合物

1

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Cat. No. Product Name Target Signaling Pathways
T10678 Carboxypeptidase G2 (CPG2) Inhibitor

CPG2 Inhibitor,Carboxypeptidase G2 Inhibitor

Carboxypeptidase Proteases/Proteasome
Carboxypeptidase G2 (CPG2) Inhibitor (CPG2 Inhibitor) 是新型的羧肽酶 G2(CPG2)抑制剂,显示出抗癌活性。
T10876 CPA inhibitor

Carboxypeptidase inhibitor

Carboxypeptidase Proteases/Proteasome
CPA inhibitor (Carboxypeptidase inhibitor) 是一种有效的羧肽酶 A (CPA) 抑制剂,Ki 值为 0.32 μM。
T3440 2-PMPA

2-(Phosphonomethyl)pentanedioic acid

Carboxypeptidase Proteases/Proteasome
2-PMPA (2-(Phosphonomethyl)pentanedioic acid) 是谷氨酸羧肽酶II 的选择性抑制剂(IC50:300 pM)。
T71126 Allixin

Allixin is a phytoallexin found in garlic (Allium sativum) bulbs. Allixin has weak antimicrobial activity and exerts an anti-promoting activity against skin tumors induced by the chemical 12-O-tetradecanoylphorbol-13-acetate (TPA). Allixin also demonstrates an inhibitory effect on aflatoxin B1-induced mutagenesis.
T16116 MLN-4760

RAAS Endocrinology/Hormones
MLN-4760 是选择性的人ACE2抑制剂,IC50=0.44 nM,对人ACE2的选择性是其他相关蛋白的 5000 多倍,包括人睾丸 ACE (IC50,>100 μM) 和牛 carboxypeptidase A (IC50,27 μM)。
T26725 AZD-9684

AZD9684,AZD 9684

AZD-9684, a carboxypeptidase U inhibitor, is used potentially for the prevention of thrombosis.
T28842 SQ-24,798

SQ 24,798,SQ24,798

SQ-24,798 is an inhibitor of the thrombin-activatable fibrinolysis and carboxypeptidase N (CPN).
T22497 2-MPPA

Others Others
glutamate carboxypeptidase II (GCP II) inhibitor
T25968 PMPA sodium

PMPA sodium salt,PMPA tetrasodium salt,PMPA Na

PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) inhibitor.
T69327 E2072

E2072 is a potent and selective thiol-based Glutamate Carboxypeptidase II (GCP-II) inhibitor.
T62423 GCPII-IN-1 TFA

GCPII-IN-1 TFA 是一种谷氨酸羧肽酶 II (GCPII; PSMA) 抑制剂支架 (Ki: 44.3 nM)。
T38420 GCPII-IN-1

GCPII-IN-1 is a potent inhibitor scaffold targeting glutamate carboxypeptidase II (GCPII), also known as prostate-specific membrane antigen (PSMA). It exhibits a high affinity for GCPII, with a binding affinity (K i ) of 44.3 nanomolar (nM).
T78239 Mergetpa

Carboxypeptidase Proteases/Proteasome
Mergetpa作为一种羧肽酶抑制剂,其功能是阻碍激肽及B2受体拮抗剂转变成无c末端精氨酸的代谢物。
T82286 Glycylglycylcysteine

Glycylglycylcysteine是一种TAFI抑制剂,其Ki值0.99μM,IC50值为9.4μM,在TAFI底物测定中有效性得以体现。TAFI为一种碱性羧肽酶,通过裂解部分降解纤维蛋白末端的赖氨酸,起到抑制纤维蛋白溶解的功能。

化合物

Carboxypeptidase G2 (CPG2) Inhibitor
Cat.No: T10678
Synonym: CPG2 Inhibitor,Carboxypeptidase G2 Inhibitor
Target: Carboxypeptidase
CPA inhibitor
Cat.No: T10876
Synonym: Carboxypeptidase inhibitor
Target: Carboxypeptidase
2-PMPA
Cat.No: T3440
Synonym: 2-(Phosphonomethyl)pentanedioic acid
Target: Carboxypeptidase
Allixin
Cat.No: T71126
Synonym:
Target:
MLN-4760
Cat.No: T16116
Synonym:
Target: RAAS
AZD-9684
Cat.No: T26725
Synonym: AZD9684,AZD 9684
Target:
SQ-24,798
Cat.No: T28842
Synonym: SQ 24,798,SQ24,798
Target:
2-MPPA
Cat.No: T22497
Synonym:
Target: Others
PMPA sodium
Cat.No: T25968
Synonym: PMPA sodium salt,PMPA tetrasodium salt,PMPA Na
Target:
E2072
Cat.No: T69327
Synonym:
Target:
GCPII-IN-1 TFA
Cat.No: T62423
Synonym:
Target:
GCPII-IN-1
Cat.No: T38420
Synonym:
Target:
Mergetpa
Cat.No: T78239
Synonym:
Target: Carboxypeptidase
Glycylglycylcysteine
Cat.No: T82286
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T8093 2-Benzylsuccinic acid

2-苄基丁二酸,DL-Benzylsuccinic acid

Carboxypeptidase Proteases/Proteasome
2-Benzylsuccinic acid (DL-Benzylsuccinic acid) 是羧肽酶 A (CPA) 抑制剂。

天然产物

2-Benzylsuccinic acid
Cat.No: T8093
Synonym: 2-苄基丁二酸,DL-Benzylsuccinic acid
Target: Carboxypeptidase
TargetMol Loading
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