14
1
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10678 |
Carboxypeptidase G2 (CPG2) Inhibitor
CPG2 Inhibitor,Carboxypeptidase G2 Inhibitor |
Carboxypeptidase | Proteases/Proteasome |
Carboxypeptidase G2 (CPG2) Inhibitor (CPG2 Inhibitor) 是新型的羧肽酶 G2(CPG2)抑制剂,显示出抗癌活性。 | |||
T10876 |
CPA inhibitor
Carboxypeptidase inhibitor |
Carboxypeptidase | Proteases/Proteasome |
CPA inhibitor (Carboxypeptidase inhibitor) 是一种有效的羧肽酶 A (CPA) 抑制剂,Ki 值为 0.32 μM。 | |||
T3440 |
2-PMPA
2-(Phosphonomethyl)pentanedioic acid |
Carboxypeptidase | Proteases/Proteasome |
2-PMPA (2-(Phosphonomethyl)pentanedioic acid) 是谷氨酸羧肽酶II 的选择性抑制剂(IC50:300 pM)。 | |||
T71126 | Allixin | ||
Allixin is a phytoallexin found in garlic (Allium sativum) bulbs. Allixin has weak antimicrobial activity and exerts an anti-promoting activity against skin tumors induced by the chemical 12-O-tetradecanoylphorbol-13-acetate (TPA). Allixin also demonstrates an inhibitory effect on aflatoxin B1-induced mutagenesis. | |||
T16116 |
MLN-4760
|
RAAS | Endocrinology/Hormones |
MLN-4760 是选择性的人ACE2抑制剂,IC50=0.44 nM,对人ACE2的选择性是其他相关蛋白的 5000 多倍,包括人睾丸 ACE (IC50,>100 μM) 和牛 carboxypeptidase A (IC50,27 μM)。 | |||
T26725 |
AZD-9684
AZD9684,AZD 9684 |
||
AZD-9684, a carboxypeptidase U inhibitor, is used potentially for the prevention of thrombosis. | |||
T28842 |
SQ-24,798
SQ 24,798,SQ24,798 |
||
SQ-24,798 is an inhibitor of the thrombin-activatable fibrinolysis and carboxypeptidase N (CPN). | |||
T22497 |
2-MPPA
|
Others | Others |
glutamate carboxypeptidase II (GCP II) inhibitor | |||
T25968 |
PMPA sodium
PMPA sodium salt,PMPA tetrasodium salt,PMPA Na |
||
PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) inhibitor. | |||
T69327 |
E2072
|
||
E2072 is a potent and selective thiol-based Glutamate Carboxypeptidase II (GCP-II) inhibitor. | |||
T62423 | GCPII-IN-1 TFA | ||
GCPII-IN-1 TFA 是一种谷氨酸羧肽酶 II (GCPII; PSMA) 抑制剂支架 (Ki: 44.3 nM)。 | |||
T38420 |
GCPII-IN-1
|
||
GCPII-IN-1 is a potent inhibitor scaffold targeting glutamate carboxypeptidase II (GCPII), also known as prostate-specific membrane antigen (PSMA). It exhibits a high affinity for GCPII, with a binding affinity (K i ) of 44.3 nanomolar (nM). | |||
T78239 |
Mergetpa
|
Carboxypeptidase | Proteases/Proteasome |
Mergetpa作为一种羧肽酶抑制剂,其功能是阻碍激肽及B2受体拮抗剂转变成无c末端精氨酸的代谢物。 | |||
T82286 |
Glycylglycylcysteine
|
||
Glycylglycylcysteine是一种TAFI抑制剂,其Ki值0.99μM,IC50值为9.4μM,在TAFI底物测定中有效性得以体现。TAFI为一种碱性羧肽酶,通过裂解部分降解纤维蛋白末端的赖氨酸,起到抑制纤维蛋白溶解的功能。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8093 |
2-Benzylsuccinic acid
2-苄基丁二酸,DL-Benzylsuccinic acid |
Carboxypeptidase | Proteases/Proteasome |
2-Benzylsuccinic acid (DL-Benzylsuccinic acid) 是羧肽酶 A (CPA) 抑制剂。 |