Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0393 |
Anastrozole
阿那曲唑,ZD1033 |
Aromatase | Endocrinology/Hormones |
Anastrozole (ZD1033) 是芳香酶的选择性抑制剂,能够抑制胎盘芳香化酶(IC50:15 nM)。 | |||
T61787 |
SYN20028567
|
||
SYN20028567, an aromatase (CYP19) inhibitor, exhibits an IC50 value of 9.4 nM. It has potential applications in breast cancer research [1]. | |||
T78590 |
Dibenzylfluorescein
DBF |
||
Dibenzylfluorescein(DBF)是一款荧光探针,作为细胞色素P450(CYP)亚型,包括CYP3A4、CYP2C8、CYP2C9、CYP2C19和CYP19的特异性底物,常在Km值0.87-1.9 µM(Ex=485nm,Em=535nm)范围内应用。该探针主要用于监测药物或疾病导致的CYP催化活性变化。 |