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4

抑制剂 & 化合物

3

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T20789	S-23 (S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide,S23	Androgen Receptor	Endocrinology/Hormones
	S-23 ((S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide) 是口服选择性雄激素受体调节剂(Ki:1.7 nM)。它能够诱导 CV-1 细胞雄激素受体介导的转录激活，提高去势大鼠前列腺、精囊和肛提肌重量。
T79088	Chlamydia pneumoniae-IN-1
	Chlamydia pneumoniae-IN-1 (compound 55)，一种抗衣原体的苯并咪唑类化合物，对肺炎衣原体具有高度抑制作用，在10 μM 浓度下能够抑制99%的肺炎衣原体生长，并对宿主细胞的活力产生95%的抑制效果。此外，Chlamydia pneumoniae-IN-1 对CV-6菌株亦显示出明显的抗菌活性，其最小抑菌浓度(MIC)为12.6 μM。
T37351	Desmethyl Bosentan
	Desmethyl bosentan is an active metabolite of the endothelin receptor antagonist bosentan .1Desmethyl bosentan (25 μM) activates the pregnane X receptor (PXR) in CV-1 monkey kidney cells expressing the human receptor in a reporter assay. 1.van Giersbergen, P.L.M., Gnerre, C., Treiber, A., et al.Bosentan, a dual endothelin receptor antagonist, activates the pregnane X nuclear receptorBr. J. Clin. Pharmacol.54(5)561-562(2002)
T36618	Rupatadine
	Rupatadine (UR-12592) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 uM(rabbit platelet membranes/guinea pig cerebellum membranes).IC50 value:Target: PAF/H1 antagonistin vitro: Rupatadine competitively inhibited histamine-induced guinea pig ileum contraction (pA2 = 9.29 +/- 0.06) without affecting contraction induced by ACh, serotonin or leukotriene D4 (LTD4). It also competitively inhibited PAF-induced platelet aggregation in washed rabbit platelets (WRP) (pA2 = 6.68 +/- 0.08) and in hu...

化合物

Cat.No: T20789

Synonym: (S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide,S23

Target: Androgen Receptor

Chlamydia pneumoniae-IN-1

Cat.No: T79088

Desmethyl Bosentan

Cat.No: T37351

Cat.No: T36618

Cat. No.	Product Name	Target	Signaling Pathways
T40718	4-Methyl-1-pentanol Isohexanol,4-甲基-1-戊醇
	4-Methyl-1-pentanol (Isohexanol) is a volatile aroma compound of red wine from cv. Kalecik Karasι.
T36738	4′-Hydroxy-2′-methylacetophenone
	4′-Hydroxy-2′-methylacetophenone, an aroma compound of red wines, is isolated from cv. Bobal grape variety. 4′-Hydroxy-2′-methylacetophenone has ciliate toxicity. 4′-Hydroxy-2′-methylacetophenone inhibits the growth of T. pyriformis, with an IC50 of 0.65 mM[1][2]. [1]. GómezGarcía-Carpintero E, et, al. Aroma characterization of red wines from cv. Bobal grape variety grown in La Mancha region. Food Research International. 2011 Jan; 44(1): 61-70. [2]. Schüürmann G, et, al. Stepwise discrimination ...
T81508	Petanin chloride
	Petanin (chloride) 为一种香豆素类花青素，源自彩色马铃薯块茎表皮。

天然产物

4-Methyl-1-pentanol

Cat.No: T40718

Synonym: Isohexanol,4-甲基-1-戊醇

4′-Hydroxy-2′-methylacetophenone

Cat.No: T36738

Petanin chloride

Cat.No: T81508

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