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Cat. No. Product Name Target Signaling Pathways
T36038 SY-5609

CDK7-IN-3

CDK Cell Cycle/Checkpoint
SY-5609 是一种选择性的非共价 CDK7 抑制剂(KD = 0.065 nM),具有抗肿瘤活性并抑制细胞凋亡。
T62926 CDK7/12-IN-1

CDK7/12-IN-1 是一种 CDK7/12 的选择性抑制剂,作用于 CDK7 (IC50: 3 nM) 和 CDK 12 (IC50: 277 nM)。抑制 CDK7CDK12 是一种有效抑制肿瘤生长的有效。
T40353 CDK7/9-IN-1

CDK7/9-IN-1

CDK7/9-IN-1 is a specific inhibitor of cyclin-dependent kinases 7/9 (CDK7/9). It specifically targets CDK7, while also displaying inhibitory activity against CDK9. CDK7/9-IN-1 demonstrates excellent inhibitory potency against CDK7, with IC50 values of 0.0656 μM and 0.00574 μM without pre-incubation and after 3 hours pre-incubation, respectively. Furthermore, CDK7/9-IN-1 inhibits CDK9 with an IC50 of 2.14 μM after 3 hours pre-incubation. Its application in cancer research makes it valuable for su...

化合物

SY-5609
Cat.No: T36038
Synonym: CDK7-IN-3
Target: CDK
CDK7/12-IN-1
Cat.No: T62926
Synonym:
Target:
CDK7/9-IN-1
Cat.No: T40353
Synonym: CDK7/9-IN-1
Target:
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