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Cat. No. Product Name Target Signaling Pathways
T36932 CD532 hydrochloride

CD532 hydrochloride is a potent inhibitor of Aurora A kinase, having an IC50 of 45 nM. It not only blocks the activity of Aurora A kinase but also facilitates the degradation of the protein MYCN. Furthermore, CD532 hydrochloride interacts directly with AURKA, inducing a significant conformational change. Its utility in cancer research has been demonstrated [1][2].
T50110 CD532

Aurora Kinase Cell Cycle/Checkpoint; Chromatin/Epigenetic
CD532 是一种高效的 Aurora A 激酶抑制剂,IC50 值为 45 nM。CD532 可阻断 Aurora A 激酶活性,驱动 MYCN 降解,可以直接与 AURKA 相互作用并诱导整体构象转变。CD532 可用于研究癌症。

化合物

CD532 hydrochloride
Cat.No: T36932
Synonym:
Target:
CD532
Cat.No: T50110
Synonym:
Target: Aurora Kinase
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