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Cat. No. Product Name Target Signaling Pathways
T9638 CCT241161

Raf MAPK
CCT241161 is an orally active pan-RAF inhibitor, with IC50 values of 3, 6, 10, 15, and 30 nM for LCK, CRAF, SRC, V600E-BRAF, and BRAF, respectively. It displays significant activity against BRAF and NRAS mutant melanomas, as well as demonstrating anticancer cell proliferative effects [1].

化合物

CCT241161
Cat.No: T9638
Synonym:
Target: Raf
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