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Cat. No. Product Name Target Signaling Pathways
T11882 Pulrodemstat benzenesulfonate

LSD1-IN-7 benzenesulfonate,CC-90011 benzenesulfonate

Histone Demethylase Chromatin/Epigenetic
Pulrodemstat benzenesulfonate (CC-90011 benzenesulfonate) 是一种有效的口服活性赖氨酸特异性去甲基化酶 1 (LSD1) 抑制剂,IC50为 0.25 nM,具有抗癌活性。它诱导急性髓细胞性白血病和小细胞肺癌细胞分化,对 LSD2、MOA-A 和 MAO-B 的酶抑制作用较小。
T39258 Pulrodemstat

LSD1-IN-7,CC-90011

Pulrodemstat (CC-90011) is a highly potent and selective inhibitor of lysine specific demethylase-1 (LSD1). It exhibits a reversible mode of action and can be administered orally. With an impressive IC50 of 0.25 nM, Pulrodemstat effectively suppresses the enzymatic activity of LSD1. Notably, it demonstrates minimal inhibition against LSD2, MOA-A, and MAO-B enzymes. Moreover, Pulrodemstat possesses remarkable anticancer properties, promoting differentiation in acute myeloid leukemia (AML) and sma...

化合物

Pulrodemstat benzenesulfonate
Cat.No: T11882
Synonym: LSD1-IN-7 benzenesulfonate,CC-90011 benzenesulfonate
Target: Histone Demethylase
Pulrodemstat
Cat.No: T39258
Synonym: LSD1-IN-7,CC-90011
Target:
TargetMol Loading
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