Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T12656 |
(Rac)-Apremilast D5
(Rac)-CC-10004 D5 |
Others | Others |
(Rac)-Apremilast D5 is a deuterium-labeled version of the enantiomer (R)-Apremilast, also known as (R)-CC-10004, which itself is one specific form of Apremilast. | |||
T10350 |
Apremilast-d5
Apremilast D5,CC-10004 D5 |
TNF; PDE | Apoptosis; Metabolism |
Apremilast D5 (CC-10004 D5) is a deuterium-labeled Apremilast. Apremilast is an orally available inhibitor of PDE-4 (IC50: 74 nM). Apremilast inhibits TNF-α release by lipopolysaccharide (IC50: 104 nM). |