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Cat. No. Product Name Target Signaling Pathways
T38287 C3a Receptor Agonist

C3a receptor agonist 1,C3a受体激动剂,Complement 3a Receptor Agonist

Complement System Immunology/Inflammation
C3a Receptor Agonist (C3a receptor agonist 1) 结合免疫系统补体途径中的G 蛋白偶联C3a 受体(C3aRs)。在肠缺血再灌注损伤模型中,C3aR 的激活可防止中性粒细胞动员。C3aRs 在成年小鼠的神经祖细胞和未成熟神经元上表达。C3a 在体外刺激神经祖细胞的分化。
T7497L1 C3a 70-77 acetate

C3a 70-77 acetate (63555-63-5 Free base)

Others Others
C3a 70-77 acetate 是对应于 C3a 的 COOH 末端的八肽乙酸酯,具有 C3a 的特异性和 1% 至 2% 的生物活性。
T7497L C3a 70-77 2TFA(63555-63-5(free base))

Complement 3a (70-77)

Complement System Immunology/Inflammation
C3a 70-77 2TFA(63555-63-5(free base)) (Complement 3a (70-77)) 是对应于 C3a 的 COOH 末端的八肽。
T7497 C3a (70-77)

Complement 3a (70-77),C3a 70-77

Complement System Immunology/Inflammation
C3a (70-77) 是对应于 C3a 的 COOH 末端的八肽。
TP1193 C3a (70-77) TFA (63555-63-5 free base)

C3a (70-77) TFA,Complement 3a (70-77) (TFA)

C3a (70-77) TFA (Complement 3a (70-77) TFA) is a COOH-terminal fragment of the C3a anaphylatoxin peptide.
T75966 C3a (70-77) (TFA)

C3a (70-77) TFA (Complement 3a (70-77) TFA) 为COOH末端对应C3a的八肽,具有C3a的特异性且生物活性约为1至2%。
T9316 JR14a

5-(Bis(4-chlorophenyl)methyl)-3-methylthiophene-2-carbonyl)-l-arginine hydrochloride

Complement System Immunology/Inflammation
JR14a (5-(Bis(4-chlorophenyl)methyl)-3-methylthiophene-2-carbonyl)-l-arginine hydrochloride) 是补体C3a 受体噻吩拮抗剂,可抑制 C3aR 介导的炎症,对人 C3a 受体的选择性高于 C5a 受体。
T12851 SB290157 trifluoroacetate

Complement System Immunology/Inflammation
SB290157 trifluoroacetate 是一种选择性 C3a 受体拮抗剂,IC50值为200 nM。
T37248 Pantothenate Kinase Inhibitor

Pantothenate Kinase Inhibitor (PANKi) is a reversible inhibitor of pantothenate kinase (PanK; IC50s = 70, 92, and 25 nM for PanK1β, PanK2, and PanK3, respectively), the rate-limiting enzyme in the synthesis of coenzyme A .1It binds to the ATP-PanK3 complex with an apparent binding constant of 300 nM and exhibits mixed-type inhibition with respect to ATP and pantothenate. PANKi inhibits CoA biosynthesis in C3A cells (IC50= 0.9 μM) with no effect on cell viability when used at concentrations up to...
T72859 11β-HSD1-IN-10

11β-HSD1-IN-10 (化合物 c3a) 是一种针对11β-HSD1的有效抑制剂,具有对人IC50值为1.8 µM。可应用于肥胖、高血糖和认知障碍研究。

化合物

C3a Receptor Agonist
Cat.No: T38287
Synonym: C3a receptor agonist 1,C3a受体激动剂,Complement 3a Receptor Agonist
Target: Complement System
C3a 70-77 acetate
Cat.No: T7497L1
Synonym: C3a 70-77 acetate (63555-63-5 Free base)
Target: Others
C3a 70-77 2TFA(63555-63-5(free base))
Cat.No: T7497L
Synonym: Complement 3a (70-77)
Target: Complement System
C3a (70-77)
Cat.No: T7497
Synonym: Complement 3a (70-77),C3a 70-77
Target: Complement System
C3a (70-77) TFA (63555-63-5 free base)
Cat.No: TP1193
Synonym: C3a (70-77) TFA,Complement 3a (70-77) (TFA)
Target:
C3a (70-77) (TFA)
Cat.No: T75966
Synonym:
Target:
JR14a
Cat.No: T9316
Synonym: 5-(Bis(4-chlorophenyl)methyl)-3-methylthiophene-2-carbonyl)-l-arginine hydrochloride
Target: Complement System
SB290157 trifluoroacetate
Cat.No: T12851
Synonym:
Target: Complement System
Pantothenate Kinase Inhibitor
Cat.No: T37248
Synonym:
Target:
11β-HSD1-IN-10
Cat.No: T72859
Synonym:
Target:
TargetMol Loading
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