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Cat. No. Product Name Target Signaling Pathways
T9634 Bomedemstat

Bomedemstat (IMG-7289) 是一种有效的,具有口服活性的且不可逆的赖氨酸特异性脱甲基酶 1 (LSD1) 抑制剂,具有表观遗传活性。Bomedemstat 具有抗癌活性,可用于急性髓性白血病 (AML) 和骨髓纤维化 (MF) 的研究。
T70008 Bomedemstat ditosylate

Bomedemstat, also known as IMG-7289, is a lysine-specific histone demethylase 1 (LSD1) inhibitor with antineoplastic activity. Bomedemstat may be useful in the treatment of acute myeloid leukaemia, myelodysplastic syndrome, and Myelofibrosis. IMG-7289 selectively inhibited proliferation and induced apoptosis of JAK2 V617F cells by concomitantly increasing expression and methylation of p53, and, independently, the pro-apoptotic factor PUMA and by decreasing the levels of its antiapoptotic antago...
T63935 Bomedemstat hydrochloride

Bomedemstat (IMG-7289) hydrochloride 是一种口服具有活力的、不可逆的 lysine-specific demethylase 1(LSD1) 抑制剂。Bomedemstat hydrochloride 能够增加 H3K4 和 H3K9 的甲基化,并改变基因表达。Bomedemstat hydrochloride 能够抑制癌细胞增殖并诱导细胞凋亡,表现出抗癌效果。
T70007 CT-179

CT-179 is a highly potent and selective small molecule inhibitor of Olig2 with excellent drug-like properties.

化合物

Bomedemstat
Cat.No: T9634
Synonym:
Target:
Bomedemstat ditosylate
Cat.No: T70008
Synonym:
Target:
Bomedemstat hydrochloride
Cat.No: T63935
Synonym:
Target:
CT-179
Cat.No: T70007
Synonym:
Target:
TargetMol Loading
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