Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T72246 |
Bicuculline methobromide
(+)-Bicuculline methobromide,d-Bicuculline methobromide,(+)-Bicuculline methobromide ; d-Bicuculline methobromide |
||
Bicuculline methobromide 是选择性GABAA 受体拮抗剂,具IC50值为3 μM。该化合物可引起哺乳类动物阵挛性强直性惊厥,且能阻断Ca2+激活的钾通道,用于癫痫等精神疾病研究。 | |||
T12043 |
(-)-Bicuculline methobromide
l-Bicuculline methobromide |
GABA Receptor | Membrane transporter/Ion channel; Neuroscience |
(-)-Bicuculline methobromide is a potent antagonist of GABAA receptor . |