Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T82914 |
Bcl-2-IN-12
|
||
Bcl-2-IN-12(Compound 1)为一高效Bcl-2抑制剂,显示IC50为6 nM,适用于癌症研究领域。 | |||
T77332 |
TV 3279
|
BCL; PKC | Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling |
TV 3279是一种新型ChE-MAI 抑制剂 ,神经保护特性取决于它们诱导抗凋亡蛋白PKC、Bcl-2、Bcl-x 和SOD 的能力,并阻止促凋亡酶甘油醛磷酸脱氢酶在PC-12和神经母细胞瘤细胞中的核易位。 | |||
T11974 | Mcl1-IN-12 | BCL | Apoptosis |
Mcl1-IN-12 has anti-tumor activity.It is a selective Mcl-1 inhibitor, less potent at Bcl-2, with Kis of 0.29 and 3.1 μM, respectively. |