Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T24644 |
Piritrexim
BW 301U |
DHFR | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism |
Piritrexim (BW 301U) 是一种可口服的脂溶性二氢叶酸还原酶抑制剂,具有肺毒性,用于研究尿路上皮癌和转移性乳腺癌。 | |||
T68684 |
Piritrexim isethionate
|
||
Piritrexim isethionate is a lipid-soluble inhibitor of dihydrofolate reductase (DHFR) that appears to be an active agent in patients with metastatic urothelial cancer when administered as a 5-day, low-dose oral schedule. |