Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5439 |
BRD4 degrader AT1
|
Epigenetic Reader Domain; PROTACs | Chromatin/Epigenetic; PROTAC |
BRD4 degrader AT1 是基于 PROTAC 技术的高选择性 Brd4 降解剂,在细胞中对 Brd4BD2 的 Kd 为 44 nM。 | |||
T13561 |
AT6
|
Others; PROTACs | Others; PROTAC |
AT6 is a PROTAC AT1 analog which is a highly selective bromodomain (Brd4) degrader. |