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Cat. No. Product Name Target Signaling Pathways
T26789 BH3I-2'

BH3I2',BH3I 2'

BH3I-2' is a cell-permeable BH3 mimetic. BH3I-2' induces apoptosis by specifically preventing BH3 domain-mediated interactions between pro-apoptotic and anti-apoptotic members of the Bcl-2 family, thereby blocking the interaction between Bcl-x and Bak BH3 by targeting the Bcl-x binding pocket.
T1493 BH3I-1

BHI1

BCL; E1/E2/E3 Enzyme Apoptosis; Ubiquitination
BH3I-1 (BHI1) 是一种Bcl-2家族拮抗剂,作用于p53/mDM2,Kd 为 5.3 μM。它抑制BakBH3 肽与Bcl-xL 结合,Ki 为 2.6 μM。

化合物

BH3I-2'
Cat.No: T26789
Synonym: BH3I2',BH3I 2'
Target:
BH3I-1
Cat.No: T1493
Synonym: BHI1
Target: BCL, E1/E2/E3 Enzyme
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