Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0211 |
Azelastine
Azelastina,Astelin,Azelastinum,氮卓斯汀 |
SARS-CoV; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience |
Azelastine (Azelastinum) 是一种选择性组胺 1 拮抗剂,可研究过敏性鼻炎、哮喘、糖尿病高脂血症和 SARS-CoV-2 。 | |||
T0211L |
Azelastine hydrochloride
Optivar,Azelastine HCl,Allergodil,盐酸氮卓斯汀,Astelin |
SARS-CoV; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience |
Azelastine hydrochloride (Astelin) 是一种选择性组胺 1拮抗剂,可研究过敏性鼻炎、哮喘、糖尿病高脂血症和 SARS-CoV-2 。 | |||
T21109 |
(S)-Azelastine hydrochloride
Azelastine hydrochloride (S)- |
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(S)-Azelastine hydrochloride, an antihistamine, has been shown to down-regulate H1R, M1R and M3R levels. It has also been shown to inhibit proliferation of HNEpC. | |||
T70675 |
(R)-Azelastine
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(R)-Azelastine is an antihistamine which has been shown to down-regulate H1R, M1R and M3R levels. This compound has also been shown to inhibit HNEpC proliferation. | |||
T70674 |
(S)-Azelastine
|
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(S)-Azelastine is an antihistamine which has been shown to down-regulate H1R, M1R and M3R levels. This compound has also been shown to inhibit HNEpC proliferation. | |||
T70481 | (R)-Azelastine hydrochloride | ||
(R)-Azelastine hydrochloride is an antihistamine which has been shown to down-regulate H1R, M1R and M3R levels. This compound has also been shown to inhibit HNEpC proliferation. | |||
T74583 |
Desmethylazelastine
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Desmethylazelastine是Azelastine经由细胞色素P450酶系统的氧化代谢形成的主要活性代谢物,具有97%的蛋白结合率和54小时的消除半衰期。Azelastine作为一种口服活性的组胺H1受体拮抗剂,特点是选择性高和亲和力强。它主要用于治疗过敏性鼻炎、哮喘、糖尿病高脂血症以及用于SARS-CoV-2的研究。 |