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Cat. No. Product Name Target Signaling Pathways
T79969 Axl-IN-16

TAM Receptor Tyrosine Kinase/Adaptors
Axl-IN-16Axl与HIF的双效抑制剂,能激发Flammulina velutipes子实体生成,并抑制HIF活性与受体酪氨酸激酶的表达。
T78834 HIV-IN-7

HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; Metabolism
Axl-IN-16(Compound 4)为Axl抑制剂,能够抑制Axl表达及抑制HIF活性,并诱导金针菇子实体形成。Axl-IN-16可通过分离红血球菌与猴头菇的“子实体液(FL)”得到。
T29062 UNC3133

UNC 3133,UNC-3133

UNC3133 is a potent and selective Mer tyrosine kinase (MerTK) inhibitor with IC50 Mer 3.0 nM; Axl 17nM; Tyro 3.31 nM; FLT3 6.6 nM; PO Cmax = 0.023; IV T1/2 = 1.59 h, %F = 16. Mer tyrosine kinase (MerTK) is aberrantly elevated in various tumor cells and ha

化合物

Axl-IN-16
Cat.No: T79969
Synonym:
Target: TAM Receptor
HIV-IN-7
Cat.No: T78834
Synonym:
Target: HIF/HIF Prolyl-Hydroxylase
UNC3133
Cat.No: T29062
Synonym: UNC 3133,UNC-3133
Target:
TargetMol Loading
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