Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T79969 |
Axl-IN-16
|
TAM Receptor | Tyrosine Kinase/Adaptors |
Axl-IN-16为Axl与HIF的双效抑制剂,能激发Flammulina velutipes子实体生成,并抑制HIF活性与受体酪氨酸激酶的表达。 | |||
T78834 |
HIV-IN-7
|
HIF/HIF Prolyl-Hydroxylase | Chromatin/Epigenetic; Metabolism |
Axl-IN-16(Compound 4)为Axl抑制剂,能够抑制Axl表达及抑制HIF活性,并诱导金针菇子实体形成。Axl-IN-16可通过分离红血球菌与猴头菇的“子实体液(FL)”得到。 | |||
T29062 |
UNC3133
UNC 3133,UNC-3133 |
||
UNC3133 is a potent and selective Mer tyrosine kinase (MerTK) inhibitor with IC50 Mer 3.0 nM; Axl 17nM; Tyro 3.31 nM; FLT3 6.6 nM; PO Cmax = 0.023; IV T1/2 = 1.59 h, %F = 16. Mer tyrosine kinase (MerTK) is aberrantly elevated in various tumor cells and ha |