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Cat. No. Product Name Target Signaling Pathways
T14349 Auristatin F

Microtubule Associated Cytoskeletal Signaling
Auristatin F 是一种有效的微管抑制剂和血管损伤剂。 Auristatin F 可用于抗体-药物偶联物。
T3256 MMAF

一甲基澳瑞他汀 F,MonoMethyl auristatin F

Others; Microtubule Associated Cytoskeletal Signaling; Others
MMAF (MonoMethyl auristatin F) 是一种抗有丝分裂剂,通过阻断微管蛋白的聚合来抑制细胞分裂,用作抗肿瘤药物和抗体偶联药物的细胞毒性成分。
T12081 MMAF-OMe

Monomethyl auristatin F methyl ester

MMAF-OMe (Monomethyl auristatin F methyl ester) 是一种抗微管蛋白剂,能够抑制 MDAMB435/5T4,MDAMB361DYT2,MDAMB468 和 Raji (5T4-) 这四种肿瘤细胞,IC50值分别为 0.056 nM,0.166 nM,0.183 nM 和 0.449 nM。它也是ADC 细胞毒素。
T18251 MAL-di-EG-Val-Cit-PAB-MMAF

Others Others
MAL-di-EG-Val-Cit-PAB-MMAF refers to a chemical compound that comprises the linker (MAL-di-EG-Val-Cit-PAB) and the potent blocker of tubulin polymerization (MMAF, Monomethyl auristatin F)[1].
T18326 MC-Val-Cit-PAB-MMAF

Others Others
MC-Val-Cit-PAB-MMAF is an antibody-drug conjugate (ADC) component that exhibits antitumor properties through the action of the tubulin inhibitor, monomethyl auristatin F (MMAF), which is connected by a cathepsin-cleavable linker, MC-Val-Cit-PAB.
T27975 MAL-PEG4-MMAF

MAL-PEG4-MMAF is a maleimido functionalized derivative of MMAF (Monomethyl auristatin F) with PEG4 linker. The maleimido functional group can be easily conjugated to protein carriers (such as antibody or enzyme). MAL-PEG4-MMAF is a useful precursor for ma
T77892 Mal-PEG8-Val-Cit-PAB-MMAF

Mal-PEG8-Val-Cit-PAB-MMAF 是一种用于抗体药物偶联体 (ADC) 的药物-连接物复合体 (drug-linker conjugate for ADC)。该化合物由一个可降解的 ADC linker 以及有效的微管蛋白抑制剂 MMAE 组成。
T77894 Val-Cit-PAB-MMAF sodium

Val-Cit-PAB-MMAFsodium为抗体药物偶联物(ADC)的活性组分,其结构由ADC连接子(肽类连接子Val-Cit-PAB)与高效微管蛋白聚合抑制剂MMAF通过偶联形成。

化合物

Auristatin F
Cat.No: T14349
Synonym:
Target: Microtubule Associated
MMAF
Cat.No: T3256
Synonym: 一甲基澳瑞他汀 F,MonoMethyl auristatin F
Target: Others, Microtubule Associated
MMAF-OMe
Cat.No: T12081
Synonym: Monomethyl auristatin F methyl ester
Target:
MAL-di-EG-Val-Cit-PAB-MMAF
Cat.No: T18251
Synonym:
Target: Others
MC-Val-Cit-PAB-MMAF
Cat.No: T18326
Synonym:
Target: Others
MAL-PEG4-MMAF
Cat.No: T27975
Synonym:
Target:
Mal-PEG8-Val-Cit-PAB-MMAF
Cat.No: T77892
Synonym:
Target:
Val-Cit-PAB-MMAF sodium
Cat.No: T77894
Synonym:
Target:
TargetMol Loading
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