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Cat. No. Product Name Target Signaling Pathways
T25107 Arginylphenylalaninamide

Rfamide,Arg-phe-NH2

Arginylphenylalaninamide, an FMRamide fragment, may be utilized as a neurotransmitter or neuromodulator by optic lobe neurons of different types.
TP2479 Sdrnflrfamide

Ser-asp-arg-asn-phe-leu-arg-phe-NH2

Sdrnflrfamide exhibits FMRFamide-like immunoreactivity isolated from the nervous system of the lobster Homarus americanus.
T31568 DP 432

DP432,beta-Alanyl-Arg-Gly-Phe-Phe-Tyr-NH2,DP-432

DP 432 is an insulin hexapeptide fragment.
TP2338 Cenupatide

UPARANT,Cenupatide trifluoroacetic acid salt,Ac-Arg-Aib-Arg-α(Me)Phe-NH2)

Cenupatide is a urokinase plasminogen activator receptor (uPAR) inhibitor. Cenupatide inhibits uPAR binding to the formyl peptide receptors (FPRs) can improve kidney lesions in a rat model of STZ-induced diabetes. Cenupatide reverted STZ-induced up-regula
T83709 LIH383 TFA

Phe-Gly-Gly-Phe-Met-Arg-Arg-Lys-NH2

LIH383是一种趋化因子(C-X-C motif) 受体7 (CXCR7)的多肽激动剂,属于趋化因子和阿片肽清除受体。它专一性激活CXCR7 (EC50 = 0.61 nM),在3 µM浓度时,相比μ-、δ-、κ-阿片受体以及诺氨酸阿片肽(NOP)受体的β-arrestin招募实验中表现出高选择性。LIH383(3 µM)通过阻止U87-ACKR3细胞中,由非选择性阿片受体激动剂dynorphin A诱导的CXCR7对阿片肽的摄取,发挥作用。
T31808 Flrlamide, manduca

Glu-asp-val-val-his-ser-phe-leu-arg-phe-Nh2,Pedvvhsflrf-NH2,Masflrfamide I

Flrlamide, manduca is a bioactive peptide extracted from the central nervous system of Manduca sexta.
T25683 Leucomyosuppressin

p-Glu-asp-val-asp-his-val-phe-leu-arg-phe-NH2

Leucomyosuppressin, isolated from head extracts of the cockroach Leucophaea maderae, inhibits evoked transmitter release at the mealworm neuromuscular junction.
TP2472 Leucopyrokinin

Pglu-thr-ser-phe-thr-pro-arg-leu-NH2

Leucopyrokinin is a myotropic neuropeptide.
T20481 Antagonist G

Arg-trp-N-methyl-phe-trp-leu-met-NH2

Antagonist G is an anticancer peptide and is also a broad spectrum neuropeptide growth factor antagonist.
T25092 Antho-rpamide II

Glu-asn-phe-his-leu-arg-pro-NH2

Antho-rpamide II is a biologically active neuropeptide isolated from the sea anemone Anthopleura elegantissima.
TP2476 Tnrnflrfamide

Thr-asn-arg-asn-phe-leu-arg-phe-NH2,Peptide F(1), lobster,F1 Peptide, lobster,Lobster peptide F1

Tnrnflrfamide is a SCP (small cardioactive peptide)-like peptide found in lobster neurons; exhibits FMRFamide-like immunoreactivity.
T32192 IRI-426

Ac-Arg-Pro-Asp-Val-Phe-NH2,IRI426

IRI-426 is a bioactive chemical.
TP2455 Locustapyrokinin II

Pglu-ser-val-pro-thr-phe-thr-pro-arg-leu-NH2

Locustapyrokinin II is a member of the FXPRL-amide peptide family isolated from Locusta migratoria.
T33516 Msh (5-10), cyclic

Cyclic H-asp-his-phe-arg-trp-lys-NH2

Msh (5-10), cyclic, as a synthetic peptide, can conjugate with fatty acids for enhanced potency.
T32400 KKI 8

N-Adamantaneacetyl-phe-arg-ser-val-gln-NH2,KKI8,KKI-8

KKI 8 is a peptide analog.
T25194 BW 443C

BW443C,BW-443C,Tyr-arg-gly-(4-nitro-phe)-pro-NH2

BW 443C is a selective agonist of mu-opioid receptor.
T32399 KKI 7

KKI-7,N-Cyclohexylacetyl-phe-arg-ser-val-gln-NH2,KKI7

KKI 7 is a peptide analog.
T24901 Troponin I (104-115)

Ac-Gly-lys-phe-lys-arg-pro-pro-leu-arg-arg-val-arg-NH2,Tni peptide (104-115)

Troponin I is a cardiac and skeletal muscle protein useful in the laboratory diagnosis of a heart attack. Troponin I is a part of the troponin protein complex, where it binds to actin in thin myofilaments to hold the actin-tropomyosin complex in place.
T25507 HP 228

HP-228,Ac-Nle-gln-his-D-phe-arg-D-trp-gly-NH2,HP228

HP 228 is a heptapeptide by inhibits the induction of nitric oxide synthase.
T25913 P-113

P 113,Ala-lys-arg-his-his-gly-tyr-lys-arg-lys-phe-his-NH2

P-113 is a peptide with antimicrobial activity.
T83666 Kisspeptin-10 (zebrafish) TFA

Tyr-Asn-Leu-Asn-Ser-Phe-Gly-Leu-Arg-Tyr-NH2,Kp-10

Kisspeptin-10是一种在斑马鱼的大脑、卵巢和睾丸中表达的神经肽,参与性腺发育和类固醇表达。在10 ng/ml的浓度下使用时,能提高孤立的斑马鱼卵巢滤泡中编码黄体生成素(luteinizing hormone, Lh)受体,以及孕酮受体a (Progestin receptor a, Pra)和Prb的mRNA水平。在0.1和1 µg/g的剂量下给予时,Kisspeptin-10能在雌性金鱼中增加黄体生成素的血清水平,但在雄性金鱼中则不会。
TP2480 Locustamyotropin

Lom-MT,Locustamyotropin I,Lom MT,LomMT,Gly-ala-val-pro-ala-ala-gln-phe-ser-pro-arg-leu-NH2

Locustamyotropin is a novel peptide isolated from Leucophae maderae; stimulates the spontaneous contractions of the hindgut of Leucophaea maderae.
T70836 DMJ-I-228

DMJ-I-228 is a specific inhibitor of HIV-1 entry through interaction with the Env spike by virtue of the incorporation of a guandinium group.
T80121 Ac-(d-Arg)-CEH-(d-Phe)-RWC-NH2

Melanocortin Receptor GPCR/G Protein; Neuroscience
Ac-DArg-c[Cys-Glu-His-DPhe-Arg-Trp-Cys]-NH2 是一种环状八肽,能够激活MC4R。该化合物能显著提高心率与血压。
T80112 Arg-Val-(Nle-p-nitro)-Phe-Glu-Ala-Nle-NH2

HIV Protease Microbiology/Virology; Proteases/Proteasome
Arg-Val-(Nle-p-nitro)-Phe-Glu-Ala-Nle-NH2 是一种用于检测HIV-1蛋白酶活性的荧光底物。
TP1095 Elamipretide

MTP-131,RX-31,SS-31

Others Others
Elamipretide (MTP-131) 是一种线粒体靶向抗氧化四肽 (D-Arg-dimethylTyr-Lys-Phe-NH2),可以减少有毒活性氧的产生并稳定心磷脂,具有血脑屏障渗透性。Elamipretide 是罕见病巴氏综合征的潜在治疗剂。
T76449 Substance P (alligator)

Substance P (alligator),一种从鳄鱼中提取的神经肽,其氨基酸序列为Arg-Pro-Arg-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2
TP1095L Elamipretide acetate

MTP 131 acetate,Elamipretide acetate (736992-21-5 Free base)

Elamipretide acetate (MTP 131 acetate) 是Elamipretide 衍生物。Elamipretide 是一种小的线粒体靶向四肽(D-Arg-dimethylTyr-Lys-Phe-NH2),可用于研究减少有毒活性氧的产生和稳定心磷脂。
T81176 Ser-parafluoroPhe-Aad-Leu-Arg-Asn-Pro-NH2

Ser-parafluoroPhe-Aad-Leu-Arg-Asn-Pro-NH2 是一种具备生物活性的肽。研究凝血酶受体束缚配体 SFLLRNP 的结构活性表明,Phe-2-苯基在受体识别过程中具有关键作用。研究还发现,将 Phe-2 替换为对氟苯丙氨酸 [(pF)Phe],可以提升其生物活性。
TP2212 a-MSH, amide

Others Others
a-MSH, amide is a peptide with the sequence Ac-Ser-Tyr-Ser-Met-Glu-His-Phe-Arg-Trp-Gly-Lys-Pro-Val-NH2, MW= 1664.9. The melanocyte-stimulating hormones (collectively referred to as MSH or intermedins) are a class of peptide hormones that are produced by c

化合物

Arginylphenylalaninamide
Cat.No: T25107
Synonym: Rfamide,Arg-phe-NH2
Target:
Sdrnflrfamide
Cat.No: TP2479
Synonym: Ser-asp-arg-asn-phe-leu-arg-phe-NH2
Target:
DP 432
Cat.No: T31568
Synonym: DP432,beta-Alanyl-Arg-Gly-Phe-Phe-Tyr-NH2,DP-432
Target:
Cenupatide
Cat.No: TP2338
Synonym: UPARANT,Cenupatide trifluoroacetic acid salt,Ac-Arg-Aib-Arg-α(Me)Phe-NH2)
Target:
LIH383 TFA
Cat.No: T83709
Synonym: Phe-Gly-Gly-Phe-Met-Arg-Arg-Lys-NH2
Target:
Flrlamide, manduca
Cat.No: T31808
Synonym: Glu-asp-val-val-his-ser-phe-leu-arg-phe-Nh2,Pedvvhsflrf-NH2,Masflrfamide I
Target:
Leucomyosuppressin
Cat.No: T25683
Synonym: p-Glu-asp-val-asp-his-val-phe-leu-arg-phe-NH2
Target:
Leucopyrokinin
Cat.No: TP2472
Synonym: Pglu-thr-ser-phe-thr-pro-arg-leu-NH2
Target:
Antagonist G
Cat.No: T20481
Synonym: Arg-trp-N-methyl-phe-trp-leu-met-NH2
Target:
Antho-rpamide II
Cat.No: T25092
Synonym: Glu-asn-phe-his-leu-arg-pro-NH2
Target:
Tnrnflrfamide
Cat.No: TP2476
Synonym: Thr-asn-arg-asn-phe-leu-arg-phe-NH2,Peptide F(1), lobster,F1 Peptide, lobster,Lobster peptide F1
Target:
IRI-426
Cat.No: T32192
Synonym: Ac-Arg-Pro-Asp-Val-Phe-NH2,IRI426
Target:
Locustapyrokinin II
Cat.No: TP2455
Synonym: Pglu-ser-val-pro-thr-phe-thr-pro-arg-leu-NH2
Target:
Msh (5-10), cyclic
Cat.No: T33516
Synonym: Cyclic H-asp-his-phe-arg-trp-lys-NH2
Target:
KKI 8
Cat.No: T32400
Synonym: N-Adamantaneacetyl-phe-arg-ser-val-gln-NH2,KKI8,KKI-8
Target:
BW 443C
Cat.No: T25194
Synonym: BW443C,BW-443C,Tyr-arg-gly-(4-nitro-phe)-pro-NH2
Target:
KKI 7
Cat.No: T32399
Synonym: KKI-7,N-Cyclohexylacetyl-phe-arg-ser-val-gln-NH2,KKI7
Target:
Troponin I (104-115)
Cat.No: T24901
Synonym: Ac-Gly-lys-phe-lys-arg-pro-pro-leu-arg-arg-val-arg-NH2,Tni peptide (104-115)
Target:
HP 228
Cat.No: T25507
Synonym: HP-228,Ac-Nle-gln-his-D-phe-arg-D-trp-gly-NH2,HP228
Target:
P-113
Cat.No: T25913
Synonym: P 113,Ala-lys-arg-his-his-gly-tyr-lys-arg-lys-phe-his-NH2
Target:
Kisspeptin-10 (zebrafish) TFA
Cat.No: T83666
Synonym: Tyr-Asn-Leu-Asn-Ser-Phe-Gly-Leu-Arg-Tyr-NH2,Kp-10
Target:
Locustamyotropin
Cat.No: TP2480
Synonym: Lom-MT,Locustamyotropin I,Lom MT,LomMT,Gly-ala-val-pro-ala-ala-gln-phe-ser-pro-arg-leu-NH2
Target:
DMJ-I-228
Cat.No: T70836
Synonym:
Target:
Ac-(d-Arg)-CEH-(d-Phe)-RWC-NH2
Cat.No: T80121
Synonym:
Target: Melanocortin Receptor
Arg-Val-(Nle-p-nitro)-Phe-Glu-Ala-Nle-NH2
Cat.No: T80112
Synonym:
Target: HIV Protease
Elamipretide
Cat.No: TP1095
Synonym: MTP-131,RX-31,SS-31
Target: Others
Substance P (alligator)
Cat.No: T76449
Synonym:
Target:
Elamipretide acetate
Cat.No: TP1095L
Synonym: MTP 131 acetate,Elamipretide acetate (736992-21-5 Free base)
Target:
Ser-parafluoroPhe-Aad-Leu-Arg-Asn-Pro-NH2
Cat.No: T81176
Synonym:
Target:
a-MSH, amide
Cat.No: TP2212
Synonym:
Target: Others
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