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3

抑制剂 & 化合物

3

天然产物

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Cat. No. Product Name Target Signaling Pathways
T36241 Arecaidine propargyl ester (hydrobromide)

Arecaidine propargyl ester is an agonist of M2muscarinic acetylcholine receptors (mAChRs).1It selectively binds to M2over M1, M3, M4, and M5mAChRs in CHO cells expressing the human receptors (Kis = 0.0871, 1.23, 0.851, 0.977, and 0.933 μM, respectively). Arecaidine propargyl ester induces contractions in isolated guinea pig atrium (pD2= 8.67). It induces apoptosis and the production of reactive oxygen species (ROS) in U87 and U251 glioblastoma cells when used at a concentration of 100 μM.2Arecai...
T22585 Arecaidine propargyl ester tosylate

Others Others
Arecaidine propargyl ester tosylate is a muscarinic receptor agonist.
T22584 Arecaidine but-2-ynyl ester tosylate

Others Others
mAChR M2 agonist

化合物

Arecaidine propargyl ester (hydrobromide)
Cat.No: T36241
Synonym:
Target:
Arecaidine propargyl ester tosylate
Cat.No: T22585
Synonym:
Target: Others
Arecaidine but-2-ynyl ester tosylate
Cat.No: T22584
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
TN1398 Arecaidine

Others Others
Arecaidine has tumorgenicity.
T5799 Arecaidine hydrochloride

Others Others
Arecaidine hydrochloride 是一种具有高效 GABA 吸收抑制功能的吡啶生物碱。它是 H+偶联的氨基酸转运蛋白 1 (PAT1,SLC36A1) 的底物,能够竞争性抑制 L-脯氨酸的摄取。
T80013 Arecaidine hydrobromide

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Arecaidine hydrobromide,一种吡啶生物碱,有效抑制GABA吸收。作为H+偶联的氨基酸转运蛋白1(PAT1,SLC36A1)的底物,它竞争性地抑制L-脯氨酸的摄取。

天然产物

Arecaidine
Cat.No: TN1398
Synonym:
Target: Others
Arecaidine hydrochloride
Cat.No: T5799
Synonym:
Target: Others
Arecaidine hydrobromide
Cat.No: T80013
Synonym:
Target: GABA Receptor
TargetMol Loading
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