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Cat. No. | Product Name | Target | Signaling Pathways |
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T36241 |
Arecaidine propargyl ester (hydrobromide)
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Arecaidine propargyl ester is an agonist of M2muscarinic acetylcholine receptors (mAChRs).1It selectively binds to M2over M1, M3, M4, and M5mAChRs in CHO cells expressing the human receptors (Kis = 0.0871, 1.23, 0.851, 0.977, and 0.933 μM, respectively). Arecaidine propargyl ester induces contractions in isolated guinea pig atrium (pD2= 8.67). It induces apoptosis and the production of reactive oxygen species (ROS) in U87 and U251 glioblastoma cells when used at a concentration of 100 μM.2Arecai... | |||
T22585 |
Arecaidine propargyl ester tosylate
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Others | Others |
Arecaidine propargyl ester tosylate is a muscarinic receptor agonist. | |||
T22584 |
Arecaidine but-2-ynyl ester tosylate
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Others | Others |
mAChR M2 agonist |
Cat. No. | Product Name | Target | Signaling Pathways |
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TN1398 | Arecaidine | Others | Others |
Arecaidine has tumorgenicity. | |||
T5799 |
Arecaidine hydrochloride
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Others | Others |
Arecaidine hydrochloride 是一种具有高效 GABA 吸收抑制功能的吡啶生物碱。它是 H+偶联的氨基酸转运蛋白 1 (PAT1,SLC36A1) 的底物,能够竞争性抑制 L-脯氨酸的摄取。 | |||
T80013 |
Arecaidine hydrobromide
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GABA Receptor | Membrane transporter/Ion channel; Neuroscience |
Arecaidine hydrobromide,一种吡啶生物碱,有效抑制GABA吸收。作为H+偶联的氨基酸转运蛋白1(PAT1,SLC36A1)的底物,它竞争性地抑制L-脯氨酸的摄取。 |