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Cat. No. Product Name Target Signaling Pathways
T10350 Apremilast-d5

Apremilast D5,CC-10004 D5

TNF; PDE Apoptosis; Metabolism
Apremilast D5 (CC-10004 D5) is a deuterium-labeled Apremilast. Apremilast is an orally available inhibitor of PDE-4 (IC50: 74 nM). Apremilast inhibits TNF-α release by lipopolysaccharide (IC50: 104 nM).
T12656 (Rac)-Apremilast D5

(Rac)-CC-10004 D5

Others Others
(Rac)-Apremilast D5 is a deuterium-labeled version of the enantiomer (R)-Apremilast, also known as (R)-CC-10004, which itself is one specific form of Apremilast.

化合物

Apremilast-d5
Cat.No: T10350
Synonym: Apremilast D5,CC-10004 D5
Target: TNF, PDE
(Rac)-Apremilast D5
Cat.No: T12656
Synonym: (Rac)-CC-10004 D5
Target: Others
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