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3

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T60555 Antiproliferative agent-3

Antiproliferative agent-3 (comp 4) 对 MCF-7 癌细胞表现出良好的活性,IC50值为 0.19 nM。
T64318 Capecitabine-2',3'-cyclic Carbonate

Others Others
Capecitabine-2',3'-cyclic Carbonate 是一种抗增殖化合物。
T2158 Nutlin-3

Nutlin3

E1/E2/E3 Enzyme Ubiquitination
Nutlin-3 是一种 MDM2 拮抗剂,抑制 MDM2-p53 相互作用 ,Ki 为 90 nM,并激活 p53

化合物

Antiproliferative agent-3
Cat.No: T60555
Synonym:
Target:
Capecitabine-2',3'-cyclic Carbonate
Cat.No: T64318
Synonym:
Target: Others
Nutlin-3
Cat.No: T2158
Synonym: Nutlin3
Target: E1/E2/E3 Enzyme
Cat. No. Product Name Target Signaling Pathways
T4S1637 gamma-Mangostin

Normangostin,γ-倒捻子素

Others; 5-HT Receptor GPCR/G Protein; Neuroscience; Others
gamma-Mangostin (Normangostin) 是从药用植物山竹的果壳中提纯的一种天然产物,是一种竞争性5-HT2A 受体拮抗剂。它是运甲状腺素蛋白原纤维化抑制剂,与甲状腺素结合位点结合并稳定了 TTR 四聚体,具有抗高血压、预防结肠癌等作用。
T14121 Actinonin

(-)-Actinonin

Aminopeptidase Metabolism
Actinonin ((-)-Actinonin) is a naturally occurring antibacterial agent produced by Actinomyces and a potent reversible peptide deformylase (PDF) inhibitor with a Ki of 0.28 nM, it also is an apoptosis inducer. Actinonin inhibits aminopeptidase M, aminopeptidase N and leucine aminopeptidase, it also inhibits MMP-1, MMP-3, MMP-8, MMP-9, and hmeprin α with Ki values of 300 nM, 1,700 nM, 190 nM, 330 nM, and 20 nM, respectively. Actinonin has antiproliferative and antitumor activities[1][2][3][4][5].

天然产物

gamma-Mangostin
Cat.No: T4S1637
Synonym: Normangostin,γ-倒捻子素
Target: Others, 5-HT Receptor
Actinonin
Cat.No: T14121
Synonym: (-)-Actinonin
Target: Aminopeptidase
TargetMol Loading
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