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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T61400 Anti-inflammatory agent 9

Anti-inflammatory agent 9 (compound 28)Anti-inflammatory agent 9 (compound 28) is a benzimidazothiazole derivative derived from tilomisole. It exhibits a higher affinity for the COX-2 enzyme compared to COX-1, thereby demonstrating promising anti-inflammatory properties. Furthermore, it demonstrates oral bioavailability [1].
T79670 Anti-inflammatory agent 56

COX Immunology/Inflammation; Neuroscience
Anti-inflammatory agent 56 (Compound 9) 是一种选择性COX-2抑制剂,IC50值为0.54 μM。该化合物展现出显著的抗氧化和抗炎效果,并能有效抑制氧化应激引起的细胞死亡。通过抑制Keap1、COX-2和iNOS,Anti-inflammatory agent 56减轻氧化应激及神经炎症。此外,其在小鼠中的急性毒性较低,LD50为1000 mg/kg。
T74954 Antimicrobial agent-9

Antimicrobial agent-9 (Compound 16) 作为一种抗菌剂,其对革兰氏阳性及革兰氏阴性细菌表现出2-8 μg/mL的最小抑菌浓度(MIC)。此外,Antimicrobial agent-9 还展现了抗炎活性。

化合物

Anti-inflammatory agent 9
Cat.No: T61400
Synonym:
Target:
Anti-inflammatory agent 56
Cat.No: T79670
Synonym:
Target: COX
Antimicrobial agent-9
Cat.No: T74954
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T83062 Anti-inflammatory agent 28

Compound 9 (Anti-inflammatory agent 28) 是一种具备肝脏保护活性的抗炎剂。

天然产物

Anti-inflammatory agent 28
Cat.No: T83062
Synonym:
Target:
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