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19

抑制剂 & 化合物

5

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Cat. No. Product Name Target Signaling Pathways
T14858 Calicheamicin

Calicheamicin γ1,卡奇霉素

Others Others
Calicheamicin (Calicheamicin γ1) 是肿瘤抗生素,可引起DNA 双链断裂,抑制DNA 合成。
T11508L Camicinal hydrochloride

GSK962040 hydrochloride

Others; Motilin Receptor GPCR/G Protein; Others
Camicinal hydrochloride (GSK962040 hydrochloride) 是胃动素受体的特异性激动剂 (pEC50 = 7.9)。
T6549 Isepamicin sulfate

Isepamicine (Isepamycin,硫酸异帕米星,Isepamicin Sulphate,Isepacin,sch21420) Sulphate

Antibacterial; Antibiotic Microbiology/Virology
Isepamicin sulfate (sch21420) Sulphate) 是一种广谱氨基糖苷类抗生素,对产生 I 型 6-乙酰转移酶的菌株具有良好的活性,通过靶向细菌 30S 核糖体亚基来抑制细菌蛋白质合成。
T12140 N-Acetyl-Calicheamicin

N-Acetyl-Calicheamicin γ,N-Acetyl-γ-calicheamicin

Antibacterial Microbiology/Virology
N-Acetyl-Calicheamicin (N-Acetyl-γ-calicheamicin)是一种具有很高抗肿瘤活性的的抗生素。
T41140 Eesperamicin A1

Eesperamicin A1

Esperamicin A1, an exceedingly potent antitumor antibiotic, is derived from Actinomadura verrucosospora cultures. This compound plays a crucial role in antitumor research.
T26123 Rosaramicin

M-4365A2 M4365A2,M 4365A2

Rosaramicin, a lipid-soluble basic macrolide, is an antibacterial substance similar to erythromycin but with a better activity against Gram-negative bacteria.
T11508 Camicinal

GSK962040

Others Others
Camicinal is a selective motilin receptor agonist (pEC50: 7.9).
T37844 Kigamicin C

Kigamicins are natural antitumor antibiotics that selectively kill pancreatic cancer PANC-1 cells only under nutrient-starved conditions. They also show antimicrobial activity against Gram-positive bacteria, including methicillin-resistant S. aureus. Kigamicin C inhibits PANC-1 cell survival in nutrient-deprived media at a 100-fold lower concentration than that required for cells maintained in nutrient-rich media. A related compound, kigamicin D, is active in vivo, suppressing the tumor growth o...
T32045 Hatomamicin

Yl 0358M A

Hatomamicin is a biochemical.
T25085 Amythiamicin B

Amythiamicin B is a novel antimicrobial antibiotic.
T26211 Sporeamicin A

SRM A,L-53-18 A,L53-18 A,L 53-18 A,SRM-A

Sporeamicin A is a new macrolide antibiotic from Saccaropolyspora.
T78047 Gemtuzumab ozogamicin

Gemtuzumab ozogamicin为抗体药物偶联物,由针对CD33单克隆抗体与Calicheamicin细胞毒性衍生物构成,用于急性髓系白血病研究。
T25447 Gentamicin

Septigen,Lyramycin,Refobacin,Centicin,Oksitselanim

Gentamicin is widely used as an antibiotic in the intensive care unit (ICU).
T40961 Lynamicin B

Lynamicin B, a promising pesticide, functions as a selective chitinase inhibitor exclusive to lepidoptera. It exhibits a Ki value of 8.76 μM, indicating its potential efficacy.
T32949 Luminamicin

Luminamicin is active against anaerobic bacteria, especially Clostridium sp.; isolated from actinomycete strain OMR-59.
T28046 Mirosamicin

A 11725 II,Antibiotic AR 5-2

Mirosamicin is a macrolide antibiotic, it has antimicrobial effect against gram-positive bacteria, some gram-negative bacteria and mycoplasma.
T28121 Mycinamicin I

Antibiotic A 11725 I,Mycinomycin I,A 11725 I

Mycinamicin I is a macrolide antibiotic.
T40662 Isepamicin

Sch 21420

Isepamicin (Sch 21420) is a potent aminoglycoside antibacterial compound with enhanced efficacy against strains harboring type I 6'-acetyltransferase. Its antibacterial spectrum encompasses Enterobacteriaceae and staphylococci, while exhibiting resistance against anaerobes, Neisseriaceae, and streptococci. Moreover, Isepamicin displays a robust concentration-dependent bactericidal effect, a prolonged post-antibiotic effect lasting several hours, and is capable of inducing adaptive resistance.
T74669 Gentamicin C1a

Gentamicin C1a,作为半合成抗生素Etimicin的前体,显示出抗菌活性,并且是Gentamicin复合物中的主要成分。

化合物

Calicheamicin
Cat.No: T14858
Synonym: Calicheamicin γ1,卡奇霉素
Target: Others
Camicinal hydrochloride
Cat.No: T11508L
Synonym: GSK962040 hydrochloride
Target: Others, Motilin Receptor
Isepamicin sulfate
Cat.No: T6549
Synonym: Isepamicine (Isepamycin,硫酸异帕米星,Isepamicin Sulphate,Isepacin,sch21420) Sulphate
Target: Antibacterial, Antibiotic
N-Acetyl-Calicheamicin
Cat.No: T12140
Synonym: N-Acetyl-Calicheamicin γ,N-Acetyl-γ-calicheamicin
Target: Antibacterial
Eesperamicin A1
Cat.No: T41140
Synonym: Eesperamicin A1
Target:
Rosaramicin
Cat.No: T26123
Synonym: M-4365A2 M4365A2,M 4365A2
Target:
Camicinal
Cat.No: T11508
Synonym: GSK962040
Target: Others
Kigamicin C
Cat.No: T37844
Synonym:
Target:
Hatomamicin
Cat.No: T32045
Synonym: Yl 0358M A
Target:
Amythiamicin B
Cat.No: T25085
Synonym:
Target:
Sporeamicin A
Cat.No: T26211
Synonym: SRM A,L-53-18 A,L53-18 A,L 53-18 A,SRM-A
Target:
Gemtuzumab ozogamicin
Cat.No: T78047
Synonym:
Target:
Gentamicin
Cat.No: T25447
Synonym: Septigen,Lyramycin,Refobacin,Centicin,Oksitselanim
Target:
Lynamicin B
Cat.No: T40961
Synonym:
Target:
Luminamicin
Cat.No: T32949
Synonym:
Target:
Mirosamicin
Cat.No: T28046
Synonym: A 11725 II,Antibiotic AR 5-2
Target:
Mycinamicin I
Cat.No: T28121
Synonym: Antibiotic A 11725 I,Mycinomycin I,A 11725 I
Target:
Isepamicin
Cat.No: T40662
Synonym: Sch 21420
Target:
Gentamicin C1a
Cat.No: T74669
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T6402 Azomycin

2-Nitroimidazole,2-硝基咪唑,Ro 05-9129,Amicin

Antibacterial; Antibiotic Microbiology/Virology
Azomycin (Ro 05-9129) 是一种可抑制有氧革兰氏阳性菌和革兰氏阴性菌的生长的抗生素。
T8257 Maduramicin ammonium

Maduramicin,Maduramycin Ammonium,马杜霉素铵盐

Apoptosis; Antibacterial; Antibiotic Apoptosis; Microbiology/Virology
Maduramicin ammonium (Maduramycin Ammonium) 是从放线菌Actinomadura rubra 中分离出来的。它是一种抗球虫药,可用于艾美耳球菌,腺苷球菌,鸡血肠球菌和分散肠球菌感染的相关研究。它诱导鸡心肌细胞凋亡。
T1326 Gentamicin sulfate

SCH9724,Gentamycin sulfate,NSC-82261,硫酸庆大霉素

ribosome; DHFR; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Gentamicin sulfate (SCH9724) 是一种广谱氨基糖苷类抗生素,用于抑制敏感生物体中的蛋白质合成。
T34611 Semduramicin

UK 61,689,Aviax,UK-61,689,UK61,689

Semduramicin is a carboxylic acid ionophore for management of chicken coccidiosis.
T34611L Semduramicin sodium

UK-61,689-2,UK 61,689-2,UK 61689-2,UK-61689-2,UK61689-2

Semduramicin sodium is a carboxylic acid ionophore for management of chicken coccidiosis.

天然产物

Azomycin
Cat.No: T6402
Synonym: 2-Nitroimidazole,2-硝基咪唑,Ro 05-9129,Amicin
Target: Antibacterial, Antibiotic
Maduramicin ammonium
Cat.No: T8257
Synonym: Maduramicin,Maduramycin Ammonium,马杜霉素铵盐
Target: Apoptosis, Antibacterial, Antibiotic
Gentamicin sulfate
Cat.No: T1326
Synonym: SCH9724,Gentamycin sulfate,NSC-82261,硫酸庆大霉素
Target: ribosome, DHFR, Antibacterial, Antibiotic
Semduramicin
Cat.No: T34611
Synonym: UK 61,689,Aviax,UK-61,689,UK61,689
Target:
Semduramicin sodium
Cat.No: T34611L
Synonym: UK-61,689-2,UK 61,689-2,UK 61689-2,UK-61689-2,UK61689-2
Target:
TargetMol Loading
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