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Cat. No. | Product Name | Target | Signaling Pathways |
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T14858 |
Calicheamicin
Calicheamicin γ1,卡奇霉素 |
Others | Others |
Calicheamicin (Calicheamicin γ1) 是肿瘤抗生素,可引起DNA 双链断裂,抑制DNA 合成。 | |||
T11508L |
Camicinal hydrochloride
GSK962040 hydrochloride |
Others; Motilin Receptor | GPCR/G Protein; Others |
Camicinal hydrochloride (GSK962040 hydrochloride) 是胃动素受体的特异性激动剂 (pEC50 = 7.9)。 | |||
T6549 |
Isepamicin sulfate
Isepamicine (Isepamycin,硫酸异帕米星,Isepamicin Sulphate,Isepacin,sch21420) Sulphate |
Antibacterial; Antibiotic | Microbiology/Virology |
Isepamicin sulfate (sch21420) Sulphate) 是一种广谱氨基糖苷类抗生素,对产生 I 型 6-乙酰转移酶的菌株具有良好的活性,通过靶向细菌 30S 核糖体亚基来抑制细菌蛋白质合成。 | |||
T12140 |
N-Acetyl-Calicheamicin
N-Acetyl-Calicheamicin γ,N-Acetyl-γ-calicheamicin |
Antibacterial | Microbiology/Virology |
N-Acetyl-Calicheamicin (N-Acetyl-γ-calicheamicin)是一种具有很高抗肿瘤活性的的抗生素。 | |||
T41140 |
Eesperamicin A1
Eesperamicin A1 |
||
Esperamicin A1, an exceedingly potent antitumor antibiotic, is derived from Actinomadura verrucosospora cultures. This compound plays a crucial role in antitumor research. | |||
T26123 |
Rosaramicin
M-4365A2 M4365A2,M 4365A2 |
||
Rosaramicin, a lipid-soluble basic macrolide, is an antibacterial substance similar to erythromycin but with a better activity against Gram-negative bacteria. | |||
T11508 |
Camicinal
GSK962040 |
Others | Others |
Camicinal is a selective motilin receptor agonist (pEC50: 7.9). | |||
T37844 |
Kigamicin C
|
||
Kigamicins are natural antitumor antibiotics that selectively kill pancreatic cancer PANC-1 cells only under nutrient-starved conditions. They also show antimicrobial activity against Gram-positive bacteria, including methicillin-resistant S. aureus. Kigamicin C inhibits PANC-1 cell survival in nutrient-deprived media at a 100-fold lower concentration than that required for cells maintained in nutrient-rich media. A related compound, kigamicin D, is active in vivo, suppressing the tumor growth o... | |||
T32045 |
Hatomamicin
Yl 0358M A |
||
Hatomamicin is a biochemical. | |||
T25085 |
Amythiamicin B
|
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Amythiamicin B is a novel antimicrobial antibiotic. | |||
T26211 |
Sporeamicin A
SRM A,L-53-18 A,L53-18 A,L 53-18 A,SRM-A |
||
Sporeamicin A is a new macrolide antibiotic from Saccaropolyspora. | |||
T78047 |
Gemtuzumab ozogamicin
|
||
Gemtuzumab ozogamicin为抗体药物偶联物,由针对CD33单克隆抗体与Calicheamicin细胞毒性衍生物构成,用于急性髓系白血病研究。 | |||
T25447 |
Gentamicin
Septigen,Lyramycin,Refobacin,Centicin,Oksitselanim |
||
Gentamicin is widely used as an antibiotic in the intensive care unit (ICU). | |||
T40961 |
Lynamicin B
|
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Lynamicin B, a promising pesticide, functions as a selective chitinase inhibitor exclusive to lepidoptera. It exhibits a Ki value of 8.76 μM, indicating its potential efficacy. | |||
T32949 |
Luminamicin
|
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Luminamicin is active against anaerobic bacteria, especially Clostridium sp.; isolated from actinomycete strain OMR-59. | |||
T28046 |
Mirosamicin
A 11725 II,Antibiotic AR 5-2 |
||
Mirosamicin is a macrolide antibiotic, it has antimicrobial effect against gram-positive bacteria, some gram-negative bacteria and mycoplasma. | |||
T28121 |
Mycinamicin I
Antibiotic A 11725 I,Mycinomycin I,A 11725 I |
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Mycinamicin I is a macrolide antibiotic. | |||
T40662 |
Isepamicin
Sch 21420 |
||
Isepamicin (Sch 21420) is a potent aminoglycoside antibacterial compound with enhanced efficacy against strains harboring type I 6'-acetyltransferase. Its antibacterial spectrum encompasses Enterobacteriaceae and staphylococci, while exhibiting resistance against anaerobes, Neisseriaceae, and streptococci. Moreover, Isepamicin displays a robust concentration-dependent bactericidal effect, a prolonged post-antibiotic effect lasting several hours, and is capable of inducing adaptive resistance. | |||
T74669 | Gentamicin C1a | ||
Gentamicin C1a,作为半合成抗生素Etimicin的前体,显示出抗菌活性,并且是Gentamicin复合物中的主要成分。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6402 |
Azomycin
2-Nitroimidazole,2-硝基咪唑,Ro 05-9129,Amicin |
Antibacterial; Antibiotic | Microbiology/Virology |
Azomycin (Ro 05-9129) 是一种可抑制有氧革兰氏阳性菌和革兰氏阴性菌的生长的抗生素。 | |||
T8257 |
Maduramicin ammonium
Maduramicin,Maduramycin Ammonium,马杜霉素铵盐 |
Apoptosis; Antibacterial; Antibiotic | Apoptosis; Microbiology/Virology |
Maduramicin ammonium (Maduramycin Ammonium) 是从放线菌Actinomadura rubra 中分离出来的。它是一种抗球虫药,可用于艾美耳球菌,腺苷球菌,鸡血肠球菌和分散肠球菌感染的相关研究。它诱导鸡心肌细胞凋亡。 | |||
T1326 |
Gentamicin sulfate
SCH9724,Gentamycin sulfate,NSC-82261,硫酸庆大霉素 |
ribosome; DHFR; Antibacterial; Antibiotic | Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology |
Gentamicin sulfate (SCH9724) 是一种广谱氨基糖苷类抗生素,用于抑制敏感生物体中的蛋白质合成。 | |||
T34611 |
Semduramicin
UK 61,689,Aviax,UK-61,689,UK61,689 |
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Semduramicin is a carboxylic acid ionophore for management of chicken coccidiosis. | |||
T34611L |
Semduramicin sodium
UK-61,689-2,UK 61,689-2,UK 61689-2,UK-61689-2,UK61689-2 |
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Semduramicin sodium is a carboxylic acid ionophore for management of chicken coccidiosis. |