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3

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T7814 Alloxan monohydrate

Proteasome Proteases/Proteasome; Ubiquitination
Alloxan Monohydrate 是一种能够引起糖尿病的致糖尿病药物。它作为蛋白酶体抑制剂,破坏胰腺中能够分泌胰岛素的B 细胞,导致实验动物患糖尿病。
T8391 Cesium chloride

氯化铯,CsCl

Potassium Channel Membrane transporter/Ion channel
Cesium chloride (CsCl) 是一种钾通道抑制剂,可以防止 Alloxan 引起的 Na+转运减少。Cesium chloride 可以诱发心律失常。
T27324 FK614

FK 614,ATx-08-001,ATx-08001,FK-614

FK-614 is a selective agonist of peroxisome proliferator-activated receptor gamma. FK-614 improves peripheral glucose utilization while decreases hepatic insulin extraction in alloxan-induced diabetic dogs.

化合物

Alloxan monohydrate
Cat.No: T7814
Synonym:
Target: Proteasome
Cesium chloride
Cat.No: T8391
Synonym: 氯化铯,CsCl
Target: Potassium Channel
FK614
Cat.No: T27324
Synonym: FK 614,ATx-08-001,ATx-08001,FK-614
Target:
Cat. No. Product Name Target Signaling Pathways
T7814L Alloxan

NSC 7169,NSC7169,NSC-7169

Alloxan is an acidic compound formed by the oxidation of URIC ACID.
TN3532 Borapetoside E

Others Others
Borapetoside E has anti-hyperglycemic activity, it can significantly reduce serum glucose levels at dose-dependent manners in alloxan-induced hyperglycemic mice and db/db type 2 diabetic mice.

天然产物

Alloxan
Cat.No: T7814L
Synonym: NSC 7169,NSC7169,NSC-7169
Target:
Borapetoside E
Cat.No: TN3532
Synonym:
Target: Others
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