38
3
Cat. No. | Product Name | Target | Signaling Pathways |
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T17387 |
Aloc-D-Ala-Phe-Lys(Aloc)-PAB-PNP
|
Others | Others |
Aloc-D-Ala-Phe-Lys(Aloc)-PAB-PNP is a cleavable linker utilized in the synthesis of antibody-drug conjugates (ADCs), which are innovative therapeutic agents that combine the targeting ability of antibodies with potent cytotoxic drugs. | |||
T31630 |
Enkephalinamide-met, ala(2)-(penta-F-phe)(4)-
|
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Enkephalinamide-met, ala(2)-(penta-F-phe)(4)- is a biochemical. | |||
T78432 |
Suc-AAPF-pNA
Suc-Ala-Ala-Pro-Phe-pNA |
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Suc-AAPF-pNA (Suc-Ala-Ala-Pro-Phe-pNA)为一种对硝基苯胺(pNA)显色底物,具备 1.7 mM 的Km值。它适用于定量分析人中性粒细胞内的游离及膜结合形式的组织蛋白酶G活性。 | |||
T34023 |
Phenylalanyl-prolyl-alanine
Phe-pro-ala |
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Phenylalanyl-prolyl-alanine is a neutral tripeptide. | |||
T34235 |
R 487
R-487,Asp-ser-phe-phe-beta-ala-leu-met-NH2,R487 |
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R 487 is a bioactive chemical. | |||
TP1261 |
Alexamorelin Met 1
(D-Mrp)-Ala-Trp-(D-Phe) |
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Alexamorelin Met 1 is one of the metabolites of alexamorelin. The heptapeptide Ala-His-D-2-methyl-Trp-Ala-Trp-D-Phe-Lys-NH2 (Alexamorelin) is a synthetic molecule which inhibits growth hormone secretagogue binding in vitro. | |||
TP2341 |
Hexapeptide-11
Peptamide 6,Fvapfp,Phe-val-ala-pro-phe-pro |
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Hexapeptide-11 is a novel proteostasis network modulator in human diploid fibroblasts. | |||
T81822 |
MeOSuc-AAPF-CMK
MeOSuc-Ala-Ala-Pro-Phe-CH₂Cl |
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MeOSuc-AAPF-CMK (MeOSuc-Ala-Ala-Pro-Phe-CH2Cl) 是蛋白酶 K 抑制剂,具有较高效能。 | |||
T32840 |
Locustakinin
Ala-phe-ser-ser-trp-gly-NH2,Lomk peptide,Locustakinn |
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Locustakinin is a myotropic peptide. | |||
TP2480 |
Locustamyotropin
Lom-MT,Locustamyotropin I,Lom MT,LomMT,Gly-ala-val-pro-ala-ala-gln-phe-ser-pro-arg-leu-NH2 |
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Locustamyotropin is a novel peptide isolated from Leucophae maderae; stimulates the spontaneous contractions of the hindgut of Leucophaea maderae. | |||
TP2478 |
WT-1 A1
Tyr-Met-Phe-Pro-agn-Ala-Pro-Tyr-Leu |
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WT-1 A1 is an attractive target for immunotherapy in patients with pancreatic adenocarcinoma. | |||
T70609 |
Bisnafide mesylate
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Bisnafide is a Naphthalimide Analogue that acts as DNA intercalator and topo II inhibitor. It is also an antiangiogenic agent. Antiangiogenic agents can normalize tumor vessels and promote the delivery of cytotoxic agents to tumor sites. | |||
T83687 |
Mca-RPPGFSAFK(Dnp)-OH TFA
(7-methoxycoumarin-4-yl)acetyl-Arg-Pro-Pro-Gly-Phe-Ser-Ala-Phe-Lys(2,4-dinitrophenyl)-OH |
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Mca-RPPGFSAFK(Dnp)-OH 是 endothelin-converting enzyme-1 (ECE-1) 的一种荧光底物。当 ECE-1 切割该底物时,会释放 7-methoxycoumarin-4-acetyl (Mca),其荧光可以用来量化 ECE-1 的活性。Mca 的激发/发射峰值分别为 328/420 nm。 | |||
T25197 |
Bz-Dab(nbd)-awfpp-nle-NH2
Bz-Dab(nbd)-ala-trp-phe-pro-pro-nle-NH2 |
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Bz-Dab(nbd)-ala-trp-phe-pro-pro-nle-NH2 is a fluorescent NK2 antagonist. | |||
TP1099 |
M-2420
Methoxycoumarin-Ser-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-Lys-dinitrophenyl |
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M-2420 is a fluorogenic substrate designed specifically for the β-secretase site found in the Swedish mutation of the amyloid precursor protein (APP). | |||
T83774 |
Shepherdin TFA
Lys-His-Ser-Ser-Gly-Cys-Ala-Phe-Leu-OH,Survivin (79-87) |
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Shepherdin是人体survivin的79-87氨基酸对应的合成肽,也是survivin与heat shock protein 90 (Hsp90)之间蛋白质-蛋白质相互作用的抑制剂。它以浓度依赖的方式与Hsp90的N末端结构域结合,并在150 µM的浓度下抑制了在分离的人源网状红细胞提取物中重组人survivin与Hsp90之间的相互作用。结合了穿膜肽penetratin或HIV Tat序列的Shepherdin肽结合物,体内外具有抗癌活性。 | |||
T83720 |
Biotin-Crosstide TFA
Biotin-Gly-Arg-Pro-Arg-Thr-Ser-Ser-Phe-Ala-Glu-Gly-OH |
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Biotin-crosstide是Akt底物crosstide的生物素化形式。 | |||
T36405 |
Pro-Adrenomedullin (153-185), human
Pro-Adrenomedullin (153-185), human,H2N-Ser-Leu-Pro-Glu-Ala-Gly-Pro-Gly-Arg-Thr-Leu-Val-Ser-Ser-Lys-Pro-Gln-Ala-His-Gly-Ala-Pro-Ala-Pro-Pro-Ser-Gly-Ser-Ala-Pro-His-Phe-Leu-OH |
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Pro-Adrenomedullin(153-185),human, (C143H224N42O43), a peptide with the sequence H2N-SLPEAGPGRTLVSSKPQAHGAPAPPSGSAPHFL-OH, MW= 3219.6. Adrenomedullin (AM) is a ubiquitously expressed peptide initially isolated from phaechromyctoma in 19931. AM was initially identified as a vasodilator, some have cited this as the most potent endogenous vasodilatory peptide found in the body2. Differences in opinion regarding the ability of AM to relax vascular tone arises from the differences in the model system... | |||
T78407 |
Suc-Ala-Ala-Phe-AMC
|
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Suc-Ala-Ala-Phe-AMC为一荧光胰凝乳蛋白酶底物,可遭肽链内切酶所水解。该化合物适用于顶体反应的体内测定及体外酶活性分析。 | |||
T25913 |
P-113
P 113,Ala-lys-arg-his-his-gly-tyr-lys-arg-lys-phe-his-NH2 |
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P-113 is a peptide with antimicrobial activity. | |||
T76621 |
Suc-Ala-Ala-Pro-Phe-SBzl
|
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Suc-Ala-Ala-Pro-Phe-SBzl 是一种化合物,可以作为大鼠小肠肥大细胞蛋白酶(RMCP I)、大鼠骨骼肌肥大细胞蛋白酶(RMCP II)和胰凝乳蛋白酶(Chymotrypsin)的底物。此外,Suc-Ala-Ala-Pro-Phe-SBzl 能够被甘氨酸(R208G)水解。 | |||
T80104 |
Z-Phe-Ala-diazomethylketone
PADK |
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Z-Phe-Ala-diazomethylketone 直接与 Aβ42 单体及其小型低聚物相结合,能抑制 Aβ42 在溶液中形成的十二聚体以及原纤维的生成,显示出在神经退行性疾病研究中的应用潜力。 | |||
T81817 |
Met-Arg-Phe-Ala
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Met-Arg-Phe-Ala为一种肽类化合物,同时作为脑啡肽生成内肽酶(EGE)的有效竞争性抑制剂,应用于神经系统疾病的研究。 | |||
T8761 |
[Leu15]-Gastrin I human
Amino Acid Sequence Glp-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Leu-Asp-Phe-NH2 |
Others | Others |
[Leu15]-Gastrin I human (Amino Acid Sequence Glp-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Leu-Asp-Phe-NH2) 基因编码人体内的蛋白质 [Leu15]-胃泌素 I。在人类染色体中,GAST 基因定位于 17q21.2。胃窦中的 G 细胞产生 [Leu15]-胃泌素 I 的前体前胃泌素。前胃泌素经过裂解和加工产生胃泌素,它对整个胃肠道上皮细胞具有营养作用。胃泌素对消化系统的生长至关重要,并刺激壁细胞产生胃酸。胃泌素通过称为胆囊收缩素(CCK) 或 CCK-B 受体 (CCK-BR) 的 G 蛋白偶联受体发挥其功能。胃泌素的释放受到食物的刺激,尤其是蛋白质饮食,并受到非常低的 pH 值的抑制。萎缩性胃炎、幽门螺杆菌感染和长期服用质子泵抑制剂感染可能导致胃泌素过度表达。胃腺癌显示高水平的胃泌素。 | |||
T76298 |
D-Ala-Gly-Phe-Met-NH2
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D-Ala-Gly-Phe-Met-NH2 是一种阿片类肽,是一种有效的阿片类 δ 受体激动剂。 | |||
T76622 |
Suc-Ala-Leu-Pro-Phe-pNA
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Suc-Ala-Leu-Pro-Phe-pNA (Suc-ALPF-pNA) 是一种 FK-506 结合蛋白 (FKBP) 的底物。 | |||
T76298L |
D-Ala-Gly-Phe-Met-NH2 monoacetate
|
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D-Ala-Gly-Phe-Met-NH2 monoacetate 是一种阿片类肽,是一种有效的阿片类 δ 受体激动剂。 | |||
T82643 |
cyclo(Phe-Ala-Gly-Arg-Arg-Arg-Gly-AEEAc)
|
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Cyclo(Phe-Ala-Gly-Arg-Arg-Arg-Gly-AEEAc) 通过抑制 GRTH/DDX25 的磷酸化,展现了其作为非激素性男性避孕药开发的潜在途径。 | |||
T80112 |
Arg-Val-(Nle-p-nitro)-Phe-Glu-Ala-Nle-NH2
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HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Arg-Val-(Nle-p-nitro)-Phe-Glu-Ala-Nle-NH2 是一种用于检测HIV-1蛋白酶活性的荧光底物。 | |||
T80191 |
His-D-beta-Nal-Ala-Trp-D-Phe-Lys-NH2 TFA
|
Endogenous Metabolite | Metabolism |
His-D-beta-Nal-Ala-Trp-D-Phe-Lys-NH2 TFA,GHRP-1的一种代谢产物,属于生长激素释放肽类。作为Ala-His-D-beta-Nal-Ala-Trp-D-Phe-Lys-NH2的同义物,GHRP-1能够刺激GH(生长激素)的释放。在大鼠垂体静态单层细胞试验中,GHRP-1可提高GH释放率和[Ca2+]i水平,但对cAMP浓度无显著影响。 | |||
T76582 |
Cys-Arg-Gly-Asp-Phe-Pro-Ala-Ser-Ser-Cys (Disulfide bridge:cys1-cys10)
|
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Cys-Arg-Gly-Asp-Phe-Pro-Ala-Ser-Ser-Cys (Disulfide bridge:cys1-cys10),为含环状RGD活性序列的十肽,作为整合素(Integrin)αIIbβ3的拮抗剂,能够抑制血小板与proMMP-13的粘附。 | |||
TP1672L |
N-Formyl-Met-Ala-Ser TFA(17351-32-5 free base)
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Others | Others |
N-Formyl-Met-Ala-Ser TFA(17351-32-5 free base) 是一种肽,与中性粒细胞上的甲酰肽受体结合。N-Formyl-Met-Ala-Ser 肽 (fMet-Ala-Ser) 与中性粒细胞上的甲酰肽受体结合。含有 N-甲酰甲硫氨酸的肽包括有效和已知的成员 N-甲酰-Met-Leu-Phe(FMLP 或 fMet-Leu-Phe)通过受体依赖性机制刺激人中性粒细胞。 | |||
T22868 | Influenza A virus fragment | Others | Others |
Influenza A virus fragment has the RNA sequence of Leu-Lys-Phe-Ala-Phe-Ser-Met-Met. | |||
TP1672 |
N-Formyl-Met-Ala-Ser
|
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N-Formyl-Met-Ala-Ser is a peptide, binds to formyl peptide receptors on neutrophils.N-Formyl-Met-Ala-Ser Peptide (fMet-Ala-Ser) binds to formyl peptide receptors on neutrophils. N-Formylmethionine-containing peptides including the most potent and known me | |||
TP2187 |
Ribosomal protein L3 peptide (202-222) amide
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Others | Others |
Ribosomal protein L3 peptide (202-222) is a peptide with the sequenceH2N-Met-Ser-His-Arg-Lys-Tyr-Glu-Ala-Pro-Arg-His-Gly-His-Leu-Gly-Phe-Leu-Pro-Arg-Lys-Arg-amide, MW=2573. | |||
TP2287 |
Rac GTPase fragment
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Others | Others |
Rac GTPase fragment is a peptide with the sequence H2N-Val-Phe-Asp-Glu-Ala-Ile-Arg-Ala-Val-OH, MW= 1019.15. Rac is a subfamily of the Rho family of GTPases, small signaling G proteins (more specifically a GTPase). | |||
TP2261 |
Interleukin II (60-70)
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Others | Others |
Interleukin II (60-70) is a peptide with the sequence NH2- LEU-THR-PHE-LYS-PHE-TYR-MET-PRO-LYS-LYS-ALA-COOH, MW= 1373.7. Interleukin 2 (IL-2) is a type of cytokine signaling molecule in the immune system, and it regulates the activities of the white blood | |||
T22800 |
Glycoprotein B (485-492)
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Others | Others |
Glycoprotein B is a peptide with the sequence H2N-Ser-Ser-Ile-Glu-Phe-Ala-Arg-Leu-OH, MW= 922.04. glycoprotein B is a viral glycoprotein that is involved in the viral cell entry of Herpes simplex virus. The herpesvirus glycoprotein B is the most highly c |
Cat. No. | Product Name | Target | Signaling Pathways |
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T20504 |
Alanylphenylalanine
NSC89630,Ala-phe,H-Ala-Phe-OH,NSC 89630,L-Alanyl-L-phenylalanine,NSC-89630 |
Endogenous Metabolite | Metabolism |
Alanylphenylalanine (Ala-phe) 是一种从小牛脑干中分离出的化合物。 | |||
T40490 |
Phenylalanylalanine
H-Phe-Ala-OH,苯并氨酰丙氨酸 |
Others | Others |
Phenylalanylalanine(H-Phe-Ala-OH)是由苯丙氨酸和丙氨酸融合形成的二肽。它在蛋白质的不完全消化或分解过程中形成[1]。 | |||
TN6428 |
Cyclo(Ala-Phe)
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Cyclo(Phe-Ala) displays significant anti-diatom activity with the inhibitory rate of 50% at the concentration of 50 microg/mL. |