Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN3367 |
Akuammidine
|
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Akuammidine shows anti-inflammatory and anti-asthmatic properties, it has opioid analgesic activity, it shows a preference for mu-opioid binding sites with Ki values of 0.6, 2.4 and 8.6 microM at mu-, delta- and kappa-opioid binding sites, respectively. | |||
TN2325 |
(Z)-Akuammidine
钩吻素丁 |
Others | Others |
(Z)-Akuammidine is a natural product | |||
TN3368 |
Akuammigine
|
Opioid Receptor; Adrenergic Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding pA2 values of 4.68. Akuammidine also shows a preference for mu-opioid binding sites with Ki val |