Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3504 |
AZD5153 6-Hydroxy-2-naphthoic acid
AZD5153,AZD5153结晶体(API形式),AZD-5153 HNT salt |
Epigenetic Reader Domain | Chromatin/Epigenetic |
AZD5153 6-Hydroxy-2-naphthoic acid (AZD5153) 是 AZD5153的6-羟基-2-萘甲酸盐形式。AZD5153是一种有口服活性的选择性 BET/BRD4溴结构域抑制剂,对BRD4的IC50值为1.7nM。 |