Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6284 |
Onalespib
AT13387,Onalespib (AT13387) |
HSP | Cytoskeletal Signaling; Metabolism |
Onalespib (AT13387) 是一种合成的、口服生物可利用的热休克蛋白 90 (Hsp90) 小分子抑制剂,Kd 值为 0.71 nM。具有潜在的抗肿瘤活性。它选择性地与 Hsp90 结合,从而抑制其伴侣功能并促进参与肿瘤细胞增殖和存活的致癌信号蛋白的降解。 | |||
T28236 |
Onalespib lactate
AT-13387 lactate,ATI-13387AU,ATI-13387,ATI 13387,ATI-13387A |
||
Onalespib lactate is a second-generation, potent and selective HSP90 Inhibitor with antitumor activity. | |||
T13387 |
Zatebradine
UL-FS-49 free base,UL-FS-49CL free base |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Zatebradine is a potent hyperpolarization-activated cyclic nucleotide-gated (HCN) channels inhibitor(IC50 of 1.96 µM). |