Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3978 |
Linerixibat
GSK2330672,Iinerixibat |
HBV | Microbiology/Virology |
Linerixibat (GSK2330672) 是高效的、不可吸收的、具有口服活性的顶端钠依赖性胆汁酸转运蛋白 (ASBT) 抑制剂,对人ASBT 的IC50为 42 nM。它是一种降脂剂,具有用于 2 型糖尿病和原发性胆源性胆管炎的研究潜力。 | |||
T28700 |
SC-435 mesylate
SC-435,SC435,SC 435 |
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SC-435 is an ileal apical sodium co-dependent bile acid transporter (ASBT). SC-435 inhibits plasma cholesterol. | |||
T70688 |
S 0960
|
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S 0960 is a dimeric bile acid analogue that acts as a specific inhibitor of the apical sodium-dependent bile salt transporter (ASBT) in the ileum. |